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المؤلفون: Daniela Giunta, Claudia Mugnaini, Maurizio Solinas, Carla Lobina, M. Paola Castelli, Alessandra Porcu
المصدر: European journal of pharmacology 791 (2016): 115–123. doi:10.1016/j.ejphar.2016.08.032
info:cnr-pdr/source/autori:Porcu A.; Lobina C.; Giunta D.; Solinas M.; Mugnaini C.; Castelli M.P./titolo:In vitro and in vivo pharmacological characterization of SSD114, a novel GABAB positive allosteric modulator/doi:10.1016%2Fj.ejphar.2016.08.032/rivista:European journal of pharmacology/anno:2016/pagina_da:115/pagina_a:123/intervallo_pagine:115–123/volume:791مصطلحات موضوعية: Male, 0301 basic medicine, Baclofen, binding, Allosteric modulator, Allosteric regulation, Stimulation, CHO Cells, GABAB receptor, Pharmacology, Mice, Reflex, Righting, 03 medical and health sciences, Cricetulus, 0302 clinical medicine, Allosteric Regulation, In vivo, Cricetinae, Animals, Positive allosteric modulator, Receptor, Baclofen-induced sedation/hypnosis, gamma-Aminobutyric Acid, Cerebral Cortex, Cyclohexylamines, Chemistry, Cell Membrane, GABA receptor antagonist, Rats, Pyrimidines, 030104 developmental biology, Receptors, GABA-B, nervous system, Competitive antagonist, 030217 neurology & neurosurgery