المؤلفون: Canale, Vittorio, Skiba-Kurek, Iwona, Klesiewicz, Karolina, Papież, Monika, Ropek, Marlena, Pomierny, Bartosz, Piska, Kamil, Koczurkiewicz-Adamczyk, Paulina, Empel, Joanna, Karczewska, Elżbieta, Zajdel, Paweł

مصطلحات موضوعية: arylsulfonamide/arylurea derivatives, biofilm eradication, multidrug-resistant staphylococcus epidermidis, tiophen, toxicophore

Relation: https://ruj.uj.edu.pl/xmlui/handle/item/327054

الاتاحة: https://ruj.uj.edu.pl/xmlui/handle/item/327054
https://doi.org/10.1021/acsmedchemlett.3c00536
https://pubs.acs.org/doi/10.1021/acsmedchemlett.3c00536

المؤلفون: Zidar, Nace, Tomašič, Tihomir, Kikelj, Danijel, Durcik, Martina, Tytgat, Jan, Peigneur, Steve, Rogers, Marc, Haworth, Alexander, Kirby, Robert W.

المصدر: European journal of medicinal chemistry, vol. 258, 115530, 2023. ; ISSN: 0223-5234

مصطلحات موضوعية: voltage-gated sodium channel, Na$_v$ channel, Na$_v$1.3, inhibitor, arylsulfonamide, acylsulfonamide, napetostno odvisni natrijev kanal, Na$_v$ kanal, zaviralci, arilsulfonamid, acilsulfonamid, nevrologija, farmacevtska kemija, info:eu-repo/classification/udc/615.4:54:616.8

وصف الملف: application/pdf; text/url

Relation: info:eu-repo/grantAgreement/ARRS//P1-0208; info:eu-repo/grantAgreement/ARRS//Z1-5458; info:eu-repo/grantAgreement/EC/FP7/245137; info:eu-repo/grantAgreement/other/F.W.O. Vlaanderen/GOC2319%20N; info:eu-repo/grantAgreement/other/F.W.O. Vlaanderen/GOA4919%20N; info:eu-repo/grantAgreement/other/F.W.O. Vlaanderen/G0E7120%20N; info:eu-repo/grantAgreement/other/KU Leuven/PDM%2F19%2F164; info:eu-repo/grantAgreement/other/F.W.O. Vlaanderen/12W7822%20N; https://repozitorij.uni-lj.si/IzpisGradiva.php?id=148297; https://repozitorij.uni-lj.si/Dokument.php?id=172387&dn=; https://repozitorij.uni-lj.si/Dokument.php?id=172386&dn=; https://plus.cobiss.net/cobiss/si/sl/bib/156075779; http://hdl.handle.net/20.500.12556/RUL-148297-4944731f-ea9d-93d7-cf75-5972bc0d0f2e

الاتاحة: https://repozitorij.uni-lj.si/IzpisGradiva.php?id=148297
https://repozitorij.uni-lj.si/Dokument.php?id=172387&dn=
https://repozitorij.uni-lj.si/Dokument.php?id=172386&dn=
https://plus.cobiss.net/cobiss/si/sl/bib/156075779
https://hdl.handle.net/20.500.12556/RUL-148297-4944731f-ea9d-93d7-cf75-5972bc0d0f2e

المؤلفون: Hausdorff, Marcel, Delpal, Adrien, Barelier, Sarah, Nicollet, Laura, Canard, Bruno, Touret, Franck, Colmant, Agathe, Coutard, Bruno, Vasseur, Jean-Jacques, Decroly, Etienne, Debart, Françoise

المساهمون: Institut des Biomolécules Max Mousseron Pôle Chimie Balard (IBMM), Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS)-Université de Montpellier (UM)-Ecole Nationale Supérieure de Chimie de Montpellier (ENSCM), Université de Montpellier (UM), Architecture et fonction des macromolécules biologiques (AFMB), Aix Marseille Université (AMU)-Centre National de la Recherche Scientifique (CNRS)-Institut National de Recherche pour l’Agriculture, l’Alimentation et l’Environnement (INRAE), Institut Hospitalier Universitaire Méditerranée Infection (IHU Marseille), ANR-20-CE11-0024,VIRAGE,Bases structurales et fonctionnelles de la methylation epitranscriptomique de genomes de virus à (+)ARN(2020)

المصدر: ISSN: 0223-5234.

مصطلحات موضوعية: 7-deaza-adenine, arylsulfonamide, bisubstrate, SARS-CoV-2, RNA cap methyltransferase, structure-guided design, [CHIM.THER]Chemical Sciences/Medicinal Chemistry

الاتاحة: https://hal.science/hal-04095336
https://hal.science/hal-04095336v1/document
https://hal.science/hal-04095336v1/file/Revised%20Manuscript%20%282%29%20F.Debart%20.pdf
https://doi.org/10.1016/j.ejmech.2023.115474

المؤلفون: Giovanna Ginestra, Teresa Gervasi, Francesca Mancuso, Federica Bucolo, Laura De Luca, Rosaria Gitto, Davide Barreca, Giuseppina Mandalari

المصدر: Microorganisms; Volume 11; Issue 6; Pages: 1522

مصطلحات موضوعية: Candida albicans, Candida glabrata, Candida parapsilosis, antifungal, arylsulfonamide, carbonic anhydrases

جغرافية الموضوع: agris

وصف الملف: application/pdf

Relation: Antimicrobial Agents and Resistance; https://dx.doi.org/10.3390/microorganisms11061522

الاتاحة: https://doi.org/10.3390/microorganisms11061522

المؤلفون: Culletta G., Allegra M., Almerico A. M., Restivo I., Tutone M.

المساهمون: Culletta G., Allegra M., Almerico A.M., Restivo I., Tutone M.

مصطلحات موضوعية: Anticancer compounds, Arylsulfonamide, Docking, Molecular dynamics, Pharmacophore modeling, Structure-based drug design, Sulfonamides, Telomerase inhibitors, Settore CHIM/08 - Chimica Farmaceutica

Relation: info:eu-repo/semantics/altIdentifier/pmid/35056139; info:eu-repo/semantics/altIdentifier/wos/WOS:000758217200001; volume:15; issue:1; firstpage:1; lastpage:21; numberofpages:21; journal:PHARMACEUTICALS; http://hdl.handle.net/10447/531996

الاتاحة: http://hdl.handle.net/10447/531996
https://doi.org/10.3390/ph15010082

المؤلفون: De Luca, Laura, Bucolo, Federica, Angeli, Andrea, Mancuso, Francesca, Crupi, Vittoria, Supuran, Claudiu T, Gitto, Rosaria

المساهمون: De Luca, Laura, Bucolo, Federica, Angeli, Andrea, Mancuso, Francesca, Crupi, Vittoria, Supuran, Claudiu T, Gitto, Rosaria

مصطلحات موضوعية: Antitumor agent, Arylsulfonamide, Carbonic anhydrase, Docking studie, Molecular modelling

وصف الملف: ELETTRONICO

Relation: info:eu-repo/semantics/altIdentifier/pmid/39278367; info:eu-repo/semantics/altIdentifier/wos/WOS:001317640900001; volume:113; firstpage:1; lastpage:6; numberofpages:6; journal:BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS; https://hdl.handle.net/11570/3316149

الاتاحة: https://hdl.handle.net/11570/3316149
https://doi.org/10.1016/j.bmcl.2024.129962

المؤلفون: Queda, Fausto, Calò, Sonia, Gwizdala, Karolina, Magalhães, João D., Cardoso, Sandra M., Chaves, Sílvia, Piemontese, Luca, Santos, M. Amélia

مصطلحات موضوعية: arylsulfonamide, donepezil, anti-neurodegeneratives, Alzheimer´s disease, AChE inhibitors, Aβ aggregation, Acetylcholinesterase, Alzheimer Disease, Amyloid beta-Peptides, Cell Line, Tumor, Cholinesterase Inhibitors, Humans, Ligands, Piperazines, Piperidines, Structure-Activity Relationship, Sulfonamides

Relation: #PLACEHOLDER_PARENT_METADATA_VALUE#; UID/QUI/00100/2013; UID/QUI/00100/ 2019; POCI-01-0145-FEDER-030712; CENTRO-01-0145-FEDER-000012; http://hdl.handle.net/10316/105262

الاتاحة: http://hdl.handle.net/10316/105262
https://doi.org/10.3390/molecules26061658

المؤلفون: Anthony J. Roecker (2283145), Mark E. Layton (1443547), Joseph E. Pero (1443532), Michael J. Kelly (1443562), Thomas J. Greshock (2178438), Richard L. Kraus (2245585), Yuxing Li (263516), Rebecca Klein (310566), Michelle Clements (3448511), Christopher Daley (1779979), Aneta Jovanovska (10906887), Jeanine E. Ballard (2413057), Deping Wang (1992346), Fuqiang Zhao (494277), Andrew P. J. Brunskill (8727768), Xuanjia Peng (8063972), Xiu Wang (591762), Haiyan Sun (201818), Andrea K. Houghton (5340860), Christopher S. Burgey (2397964)

مصطلحات موضوعية: Biochemistry, Medicine, Genetics, Molecular Biology, Pharmacology, Biotechnology, Sociology, Cancer, Hematology, Infectious Diseases, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, target modulation, compound 19, Lead optimization efforts, side effects, Selectivity Profile, Na v 1.7 electrophysiology protocols, novel multiparameter optimization, Na v 1.6, Na v 1.5, novel series, IVIVC, arylsulfonamide Na v 1.7 inhibitors, pain afflictions, vivo correlations, side effects preclinically, MPO Methods, target selectivity profile, voltage-gated sodium channel Na v 1.7

Relation: https://figshare.com/articles/journal_contribution/Discovery_of_Arylsulfonamide_Na_sub_v_sub_1_7_Inhibitors_IVIVC_MPO_Methods_and_Optimization_of_Selectivity_Profile/14714148

الاتاحة: https://doi.org/10.1021/acsmedchemlett.1c00218.s002

المؤلفون: Inês C. Santos (10271875), Jennifer S. Brodbelt (1308045)

مصطلحات موضوعية: Biophysics, Biochemistry, Molecular Biology, Pharmacology, Biotechnology, Environmental Sciences not elsewhere classified, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, binding affinities, mass spectrometry-based strategies, arylsulfonamide inhibitors, UVPD, carbon dioxide, mass spectrometry, ligand binding, hCAII, protein sequence, interaction, protein conformations, Carbonic anhydrase, ion mobility, Ultraviolet Photodissociation Mass ., charge states, Structural Characterization, supercharging agent, complex, binding cavity, fragmentation patterns, carbonic anhydrase II

Relation: https://figshare.com/articles/journal_contribution/Structural_Characterization_of_Carbonic_Anhydrase_Arylsulfonamide_Complexes_Using_Ultraviolet_Photodissociation_Mass_Spectrometry/14182786

الاتاحة: https://doi.org/10.1021/jasms.1c00004.s001

المؤلفون: Santamaria, S, Buemi, F, Nuti, E, Cuffaro, D, De Vita, E, Tuccinardi, T, Rossello, A, Howell, S, Mehmood, S, Snijders, AP, De Groot, R

المساهمون: British Heart Foundation

مصطلحات موضوعية: Science & Technology, Life Sciences & Biomedicine, Biochemistry & Molecular Biology, Chemistry, Medicinal, Pharmacology & Pharmacy, ADAMTS-7, ADAMTS7, activity assay, inhibitor, coronary artery disease, ARYLSULFONAMIDE INHIBITORS, CLEAVAGE, DOMAIN, AGGRECAN, BINDING, SITE, Medicinal & Biomolecular Chemistry, 0304 Medicinal and Biomolecular Chemistry, 0601 Biochemistry and Cell Biology

Relation: Journal of Enzyme Inhibition and Medicinal Chemistry; http://hdl.handle.net/10044/1/92315; FS/IBSRF/20/25032; PG/18/19/33584

الاتاحة: http://hdl.handle.net/10044/1/92315
https://doi.org/10.1080/14756366.2021.1983808

المؤلفون: Lena Cook, Tiziano Tuccinardi, Caterina Camodeca, Armando Rossello, Tanja Kellermann, Elisa Nuti, Doretta Cuffaro, Lidia Ciccone, Jörg W. Bartsch

المصدر: ACS Medicinal Chemistry Letters

مصطلحات موضوعية: ADAM8 dimerization, bifunctional inhibitors, arylsulfonamide hydroxamates, anticancer drugs, bifunctional inhibitors, anticancer drugs, Letter, Stereochemistry, Chemistry, Organic Chemistry, Drug Discovery, ADAM8 dimerization, arylsulfonamide hydroxamates, Biochemistry, ADAM8

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cf3aaed63a6f7249101b38beaedca8ec
http://europepmc.org/articles/PMC8805605

المؤلفون: Cuffaro, Doretta, Nuti, Elisa, Gifford, Valentina, Ito, Noriko, Camodeca, Caterina, Tuccinardi, Tiziano, Nencetti, Susanna, Orlandini, Elisabetta, Itoh, Yoshifumi, Rossello, Armando

المساهمون: Cuffaro, Doretta, Nuti, Elisa, Gifford, Valentina, Ito, Noriko, Camodeca, Caterina, Tuccinardi, Tiziano, Nencetti, Susanna, Orlandini, Elisabetta, Itoh, Yoshifumi, Rossello, Armando

مصطلحات موضوعية: Arylsulfonamide hydroxamate, Bifunctional inhibitor, MMP inhibitor, MT1-MMP homodimerization, Biochemistry, Molecular Medicine, Molecular Biology, Drug Discovery3003 Pharmaceutical Science, Clinical Biochemistry, Organic Chemistry

Time: 3003

وصف الملف: ELETTRONICO

Relation: info:eu-repo/semantics/altIdentifier/pmid/30522899; info:eu-repo/semantics/altIdentifier/wos/WOS:000453233300020; volume:27; issue:1; firstpage:196; lastpage:207; numberofpages:12; journal:BIOORGANIC & MEDICINAL CHEMISTRY; http://hdl.handle.net/11568/938174; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85057829887; http://www.journals.elsevier.com/bioorganic-and-medicinal-chemistry/

الاتاحة: http://hdl.handle.net/11568/938174
https://doi.org/10.1016/j.bmc.2018.11.041
http://www.journals.elsevier.com/bioorganic-and-medicinal-chemistry/

المؤلفون: Mersal, Karim I., Abdel-Maksoud, Mohammed S., Ali, Eslam M.H., Ammar, Usama M., Zaraei, Seyed-Omar, Haque, Md Mamunul, Das, Tanuza, Hassan, Noha F., Kim, Eunice EunKyeong, Lee, Jun-Seok, Park, HaJeung, Lee, Kwan Hyi, El-Gamal, Mohammed I., Kim, Hee-Kwon, Ibrahim, Tamer M., Oh, Chang-Hyun

مصطلحات موضوعية: Arylsulfonamide, Cancer, JNK, Leukemia, Pyrazole

Relation: https://napier-repository.worktribe.com/file/3198043/1/Evaluation%20of%20novel%20pyrazol-4-yl%20pyridine%20derivatives%20possessing%20arylsulfonamide%20tethers%20as%20c-Jun%20N-terminal%20kinase%20%28JNK%29%20inhibitors%20in%20leukemia%20cells

الاتاحة: https://doi.org/10.1016/j.ejmech.2023.115779
https://napier-repository.worktribe.com/file/3198043/1/Evaluation%20of%20novel%20pyrazol-4-yl%20pyridine%20derivatives%20possessing%20arylsulfonamide%20tethers%20as%20c-Jun%20N-terminal%20kinase%20%28JNK%29%20inhibitors%20in%20leukemia%20cells

المؤلفون: Hausdorff, M., Delpal, A., Barelier, S., Nicollet, L., Canard, B., Touret, F., /Colmant, Agathe, Coutard, B., Vasseur, J. J., Decroly, E., Debart, F.

مصطلحات موضوعية: 7-deaza-adenine, Arylsulfonamide, Bisubstrate, SARS-CoV-2, RNA cap, Methyltransferase, Structure -guided design

Relation: https://www.documentation.ird.fr/hor/fdi:010088101; oai:ird.fr:fdi:010088101; Hausdorff M., Delpal A., Barelier S., Nicollet L., Canard B., Touret F., Colmant Agathe, Coutard B., Vasseur J. J., Decroly E., Debart F. Structure-guided optimization of adenosine mimetics as selective and potent inhibitors of coronavirus nsp14 N7-methyltransferases. 2023, 256, p. 115474 [19 p.]

الاتاحة: https://www.documentation.ird.fr/hor/fdi:010088101

المؤلفون: Pirnat, Živa

المساهمون: Zidar, Nace

مصطلحات موضوعية: inhibitor, Nav1.3, napetostno odvisni natrijevi kanalčki, protibolečinsko sredstvo, voltage-dependent sodium channels, zaviralec, analgesic, arylsulfonamide, arilsulfonamid

وصف الملف: application/pdf

URL الوصول: https://explore.openaire.eu/search/publication?articleId=od______3505::3ed1542fa399db87f6dd84922aa3ac01
https://repozitorij.uni-lj.si/Dokument.php?id=164921&dn=

المؤلفون: Kourghi, M., De Ieso, M., Nourmohammadi, S., Pei, J., Yool, A.

المصدر: http://dx.doi.org/10.3389/fchem.2018.00142.

مصطلحات موضوعية: major intrinsic protein, MIP, AQP1, water channel, non-selective cation channel, cyclic GMP, arylsulfonamide

وصف الملف: application/pdf

Relation: http://purl.org/au-research/grants/arc/DP160104641; Frontiers in Chemistry, 2018; 6(APR):142-1-142-12; http://hdl.handle.net/2440/112299; De Ieso, M. [0000-0002-2402-4483]; Nourmohammadi, S. [0000-0002-9469-2874]; Pei, J. [0000-0003-2453-929X]; Yool, A. [0000-0003-1283-585X]

الاتاحة: http://hdl.handle.net/2440/112299
https://doi.org/10.3389/fchem.2018.00142

المؤلفون: Elena De Vita, Frederic Buemi, Shahid Mehmood, Rens de Groot, Salvatore Santamaria, Ambrosius P. Snijders, Elisa Nuti, Doretta Cuffaro, Tiziano Tuccinardi, Armando Rossello, Steven Howell

المساهمون: British Heart Foundation

المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry
article-version (VoR) Version of Record
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 36, Iss 1, Pp 2160-2169 (2021)

مصطلحات موضوعية: ADAMTS7, Endogeny, Chemistry, Medicinal, 0601 Biochemistry and Cell Biology, Substrate Specificity, DOMAIN, ADAMTS-7, Drug Discovery, BINDING, Fluorescence Resonance Energy Transfer, Pharmacology & Pharmacy, Chemical Biology & High Throughput, Molecular Structure, Chemistry, ADAMTS, SITE, General Medicine, activity assay, inhibitor, Biochemistry, Life Sciences & Biomedicine, coronary artery disease, Research Article, Research Paper, Biochemistry & Molecular Biology, Extracellular protease, High-throughput screening, Medicinal & Biomolecular Chemistry, ADAMTS7 Protein, RM1-950, Biochemistry & Proteomics, Structure-Activity Relationship, Drug Development, Ic50 values, Humans, Chelation, Protease Inhibitors, Computational & Systems Biology, Fluorescent Dyes, Pharmacology, Science & Technology, Dose-Response Relationship, Drug, 0304 Medicinal and Biomolecular Chemistry, CLEAVAGE, AGGRECAN, Substrate (chemistry), ARYLSULFONAMIDE INHIBITORS, Förster resonance energy transfer, Therapeutics. Pharmacology

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6e5ff67fe2a08544459c87feed5469a4

المؤلفون: Pirnat, Živa

المساهمون: Zidar, Nace

مصطلحات موضوعية: arilsulfonamid, napetostno odvisni natrijevi kanalčki, Nav1.3, protibolečinsko sredstvo, zaviralec, analgesic, arylsulfonamide, inhibitor, voltage-dependent sodium channels

وصف الملف: application/pdf

Relation: https://repozitorij.uni-lj.si/IzpisGradiva.php?id=143292; https://repozitorij.uni-lj.si/Dokument.php?id=164921&dn=; http://hdl.handle.net/20.500.12556/RUL-143292

الاتاحة: https://repozitorij.uni-lj.si/IzpisGradiva.php?id=143292
https://repozitorij.uni-lj.si/Dokument.php?id=164921&dn=
https://hdl.handle.net/20.500.12556/RUL-143292

المؤلفون: Shiow Lin Pan, Tsui Chin Huang, Ya Wen Cheng, Han Li Huang, Yi Min Liu, Ting Yi Sung, Jing Ping Liou

المصدر: Theranostics

مصطلحات موضوعية: Male, 0301 basic medicine, Indoles, TIMP3, Angiogenesis, Mice, Nude, Medicine (miscellaneous), Angiogenesis Inhibitors, Antineoplastic Agents, colorectal cancer, Kaplan-Meier Estimate, Matrix metalloproteinase, MPT0B390, Metastasis, 03 medical and health sciences, 0302 clinical medicine, Cell Movement, In vivo, Cell Line, Tumor, Biomarkers, Tumor, medicine, Animals, Humans, Enhancer of Zeste Homolog 2 Protein, Arylsulfonates, Neoplasm Metastasis, Promoter Regions, Genetic, Pharmacology, Toxicology and Pharmaceutics (miscellaneous), Aged, Tissue Inhibitor of Metalloproteinase-3, Migration Assay, Cell growth, Chemistry, Cell migration, Middle Aged, Prognosis, medicine.disease, Xenograft Model Antitumor Assays, Urokinase receptor, 030104 developmental biology, 030220 oncology & carcinogenesis, arylsulfonamide inducer, Cancer research, Female, Erratum, Colorectal Neoplasms, Research Paper

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7bd1ed7d47b3d31f1d74d85963885a5a
http://europepmc.org/articles/PMC6771239

المؤلفون: Sandra M. Cardoso, M. Amélia Santos, Fausto Queda, Sonia Calò, Sílvia Chaves, Luca Piemontese, Karolina Gwizdala, João D. Magalhães

المصدر: Molecules
Volume 26
Issue 6
Molecules, Vol 26, Iss 1658, p 1658 (2021)

مصطلحات موضوعية: Drug, Aβ aggregation, Alzheimer´s disease, media_common.quotation_subject, Pharmaceutical Science, Pharmacology, AChE inhibitors, Ligands, Article, Piperazines, Analytical Chemistry, lcsh:QD241-441, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, 0302 clinical medicine, lcsh:Organic chemistry, Piperidines, Alzheimer Disease, Cell Line, Tumor, Drug Discovery, medicine, Humans, Physical and Theoretical Chemistry, arylsulfonamide, Donepezil, IC50, 030304 developmental biology, media_common, 0303 health sciences, Sulfonamides, Amyloid beta-Peptides, Chemistry, Drug discovery, Organic Chemistry, Biological activity, Acetylcholinesterase, donepezil, Chemistry (miscellaneous), Molecular Medicine, anti-neurodegeneratives, Cholinesterase Inhibitors, Pharmacophore, Lead compound, 030217 neurology & neurosurgery, medicine.drug

وصف الملف: application/pdf

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d27c64ffc7590e3ff302a2328c2e11fe
http://europepmc.org/articles/PMC8002323