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1Academic Journal
المؤلفون: Anthony J. Salerno, Zhiqing He, Annika Goos-nilsson, Harri Ahola, Paul Mak
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.328.6360; http://nar.oxfordjournals.org/content/24/4/566.full.pdf
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المؤلفون: Martin Hegen, David C. Wood, Patrik Rhönnstad, Felix Vajdos, Atli Thorarensen, Mark E. Schnute, Timothy Braden, Kimberly Crouse, Maria Sjöberg, John I. Trujillo, Ravi G. Kurumbail, Bolette Husman, Konrad F. Koehler, Mattias Wennerstål, Tomas Bonn, Joakim Löfstedt, Eva Backström-Rydin, Bo Carlsson, Aron Sundell, Ming Z. Chen, Steven E. Heasley, John David Trzupek, Annika Goos-Nilsson, Carol A. Menard, Peter Harris, James R. Kiefer, Martin Bengtsson, Leon P. Collis, Michael J. Prinsen, Philippe Nuhant, Jennifer Alley, Scott A. Long, Alexander E. Hromockyj, Andrew C. Flick, Johnny Sandberg, Christoph W. Zapf, Edouard Zamaratski, Xiao Hu, Lee Napierata, Björn Kauppi, Nicole Caspers, Kimberly F. Fennell, Robert E. Kyne, Gabriel Berstein, Neelu Kaila, Lars Kruger, Wei Li, Li Xing, Ray Unwalla, Elisabet Kallin, Matthew J. Pelc, Susan Fish, James Robert Blinn, Hjalmar Gullberg, Marvin J. Meyers, Scot Richard Mente, Chulho Choi, Falgun Shah, Mathias Färnegårdh, Dean Messing, Peter G. Jones, Yajuan Zhao, Alexandria P. Taylor, Maria Sandström, Charles W. Bolten, Daniel Nöteberg, Robin A. Weinberg, Tomasz Janosik, John D. Knafels, Anna Wilhelmsson
المصدر: Journal of medicinal chemistry. 61(23)
مصطلحات موضوعية: 0301 basic medicine, Drug Inverse Agonism, Stereochemistry, Pyridines, Retinoic acid, Drug Evaluation, Preclinical, Administration, Oral, Biological Availability, 01 natural sciences, 03 medical and health sciences, chemistry.chemical_compound, Mice, RAR-related orphan receptor gamma, Drug Discovery, Inverse agonist, Animals, Humans, Benzamide, Receptor, Orphan receptor, 010405 organic chemistry, Nuclear Receptor Subfamily 1, Group F, Member 3, 0104 chemical sciences, Retinoic acid receptor, 030104 developmental biology, chemistry, Nuclear receptor, Drug Design, Molecular Medicine, Th17 Cells
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المؤلفون: Baihua Hu, Elaine Quinet, Irene Feingold, Igor Goljer, Thomas J. Berrodin, Mark J. Evans, James W Jetter, Jay Wrobel, Rayomand J. Unwalla, Michael D Basso, Annika Goos Nilsson, Anna Wilhelmsson
المصدر: Journal of Medicinal Chemistry. 53:3296-3304
مصطلحات موضوعية: Male, Models, Molecular, Transcriptional Activation, Agonist, Duodenum, medicine.drug_class, Pharmacology, Kidney, Cell Line, Sulfone, Mice, Radioligand Assay, Structure-Activity Relationship, chemistry.chemical_compound, Quinoxaline, Quinoxalines, Drug Discovery, Coactivator, medicine, Animals, Humans, Structure–activity relationship, Sulfones, Liver X receptor, Triglycerides, Liver X Receptors, Mice, Knockout, Chemistry, Kidney metabolism, Atherosclerosis, Orphan Nuclear Receptors, Mice, Inbred C57BL, Cholesterol, Liver, Biochemistry, Organ Specificity, Cell culture, Area Under Curve, Molecular Medicine, ATP-Binding Cassette Transporters, lipids (amino acids, peptides, and proteins), ATP Binding Cassette Transporter 1, Half-Life
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المؤلفون: Baihua Hu, Rayomand J. Unwalla, Mark J. Evans, Jay E. Wrobel, Annika Goos-Nilsson, Anna Wilhelmsson, Michael D. Collini, Irene Feingold, Ron Bernotas, Ponnal Nambi, Elaine Quinet
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:689-693
مصطلحات موضوعية: Agonist, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Blood–brain barrier, Biochemistry, Cell Line, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Computer Simulation, Sulfones, Liver X receptor, Molecular Biology, Binding selectivity, Liver X Receptors, Binding Sites, Organic Chemistry, Quinoline, Hydrogen Bonding, Quinoline analog, Orphan Nuclear Receptors, Rats, medicine.anatomical_structure, Nuclear receptor, chemistry, Blood-Brain Barrier, Quinolines, Molecular Medicine, ATP-Binding Cassette Transporters, ATP Binding Cassette Transporter 1, Protein Binding
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المؤلفون: Christine Huselton, David H. Kaufman, Annika Goos-Nilsson, Jay E. Wrobel, Irene Feingold, Ponnal Nambi, Ronald C. Bernotas, Elaine Quinet, Anna Wilhelmsson, Jeremy M. Travins
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:526-530
مصطلحات موضوعية: Agonist, Benzimidazole, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Cell Line, Sulfone, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, polycyclic compounds, medicine, Animals, Humans, Potency, Structure–activity relationship, RNA, Messenger, Sulfones, Liver X receptor, Molecular Biology, Liver X Receptors, Chemistry, Organic Chemistry, Biological activity, Orphan Nuclear Receptors, Rats, Microsomes, Liver, Microsome, Molecular Medicine, ATP-Binding Cassette Transporters, Benzimidazoles, lipids (amino acids, peptides, and proteins)
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المؤلفون: Anna Wilhelmsson, Ronald C. Bernotas, David H. Kaufman, Rayomand J. Unwalla, Elaine Quinet, John W. Ullrich, Annika Goos-Nilsson, Ponnal Nambi, Robert R. Singhaus, Jay E. Wrobel
المصدر: Bioorganic & Medicinal Chemistry. 17:8086-8092
مصطلحات موضوعية: Models, Molecular, Agonist, Magnetic Resonance Spectroscopy, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Ether, Alcohol, Binding, Competitive, Biochemistry, Mass Spectrometry, Cell Line, Mice, chemistry.chemical_compound, Amide, Drug Discovery, polycyclic compounds, medicine, Animals, Liver X receptor, Molecular Biology, Liver X Receptors, Macrophages, Aryl, Organic Chemistry, Quinoline, food and beverages, Orphan Nuclear Receptors, chemistry, Nuclear receptor, Alcohols, Quinolines, Molecular Medicine, lipids (amino acids, peptides, and proteins)
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المؤلفون: Elaine Quinet, Baihua Hu, Jay E. Wrobel, Anna Wihelmsson, Ponnal Nambi, Raymound Unwalla, Michael D. Collini, Annika Goos-Nilsson, Irene Feingold
المصدر: Bioorganic & Medicinal Chemistry. 17:3519-3527
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Receptors, Cytoplasmic and Nuclear, Pharmaceutical Science, Heterocyclic Compounds, 2-Ring, Biochemistry, Cell Line, Mice, Structure-Activity Relationship, Drug Discovery, Animals, Humans, Moiety, Computer Simulation, Binding site, Liver X receptor, Molecular Biology, Binding selectivity, Liver X Receptors, Chemistry, Liver cell, Organic Chemistry, Orphan Nuclear Receptors, DNA-Binding Proteins, Nuclear receptor, Cell culture, Quinolines, Molecular Medicine, ATP-Binding Cassette Transporters, Signal transduction, Sterol Regulatory Element Binding Protein 1, ATP Binding Cassette Transporter 1
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المؤلفون: Peer B. Jacobson, Lars Öhman, Birgitta Gelius, Marlena Grynfarb, Annika Goos-Nilsson, Richards Steven J, Masha Kalmanovich, Steven Fung, Thomas W. von Geldern, Denise Wilcox, Marie K. Österlund, Phong Nguyen, Jiahong Wang
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:6086-6090
مصطلحات موضوعية: medicine.drug_class, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Steroid, Bile Acids and Salts, Structure-Activity Relationship, chemistry.chemical_compound, Receptors, Glucocorticoid, fluids and secretions, Glucocorticoid receptor, In vivo, Microsomes, Drug Discovery, polycyclic compounds, medicine, Animals, Humans, Molecular Biology, Molecular Structure, Bile acid, Chemistry, Organic Chemistry, Cholic acid, Biological activity, Mifepristone, Rats, Molecular Medicine, Glucocorticoid, medicine.drug
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المؤلفون: Liang Chen, Ponnal Nambi, Qiang-Yuan Liu, Rayomand J Unwalla, Valerie Clerin, Michael D Basso, Mathias Färnegårdh, Irene Feingold, Dawn A. Savio, James Carl Keith, Christopher P. Miller, Jay Wrobel, Anita R Halpern, Farooq Azam, Anna Wilhelmsson, Annika Goos-Nilsson, Robert R. Singhaus, Christine Resmini, Christine Huselton, Baihua Hu, Michael D. Collini, Elaine M. Quinet, Tomas Bonn, Cristofer Enroth
المصدر: Journal of Medicinal Chemistry. 49:6151-6154
مصطلحات موضوعية: Male, Models, Molecular, Transcriptional Activation, Biological Availability, Receptors, Cytoplasmic and Nuclear, In Vitro Techniques, Ligands, Cell Line, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Transactivation, Drug Stability, In vivo, Drug Discovery, Animals, Humans, Structure–activity relationship, Liver X receptor, Liver X Receptors, Phenylacetates, Binding Sites, Molecular Structure, biology, Anticholesteremic Agents, Quinoline, Biological activity, Atherosclerosis, Orphan Nuclear Receptors, Protein Structure, Tertiary, DNA-Binding Proteins, Mice, Inbred C57BL, Cholesterol, chemistry, Biochemistry, ABCA1, LDL receptor, Microsomes, Liver, Quinolines, biology.protein, Molecular Medicine, ATP-Binding Cassette Transporters, Female, lipids (amino acids, peptides, and proteins), ATP Binding Cassette Transporter 1
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المؤلفون: Phong Nguyen, Sue J. Swanson, Jyoti R. Patel, Jiahong Wang, Annika Goos-Nilsson, J.T. Link, Peer B. Jacobson, Zhenping Tian, Marlena Grynfarb, Jia Du, James M. Schmidt, Brad Zinker, Thomas W von Geldern, Steven Fung, Thomas J Reisch, Denise Wilcox, Gary Rotert, Benjamin C. Lane, Bach Hickman, Bryan Sorensen
المصدر: Journal of Medicinal Chemistry. 48:5295-5304
مصطلحات موضوعية: Male, Transcriptional Activation, Benzylamines, Hypothalamo-Hypophyseal System, medicine.medical_specialty, Side effect, Pituitary-Adrenal System, Dexamethasone, Rats, Sprague-Dawley, Mice, Radioligand Assay, chemistry.chemical_compound, Cricetulus, Receptors, Glucocorticoid, Glucocorticoid receptor, Genes, Reporter, Pregnancy, Cricetinae, Internal medicine, Drug Discovery, medicine, Animals, Humans, Hypoglycemic Agents, Receptor, Glucocorticoids, Cells, Cultured, Tyrosine Transaminase, chemistry.chemical_classification, Sulfonamides, Triglyceride, Cholesterol, Uterus, Fatty acid, Alkaline Phosphatase, Rats, medicine.anatomical_structure, Endocrinology, chemistry, Hepatocytes, Molecular Medicine, Female, Antagonism, Hypothalamic–pituitary–adrenal axis
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المؤلفون: Marlena Grynfarb, Maurice Emery, J.T. Link, Noah Tu, Bryan K. Sorensen, Bach Nguyen, Annika Goos-Nilsson
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:4179-4183
مصطلحات موضوعية: medicine.drug_class, medicine.medical_treatment, Clinical Biochemistry, Biological Availability, Pharmaceutical Science, Biochemistry, Chemical synthesis, Steroid, Bile Acids and Salts, Rats, Sprague-Dawley, Receptors, Glucocorticoid, Glucocorticoid receptor, Pharmacokinetics, Drug Discovery, medicine, Animals, Potency, Receptor, Molecular Biology, Bile acid, Chemistry, Organic Chemistry, Ligand (biochemistry), Rats, Molecular Medicine
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المؤلفون: Marlena Grynfarb, Maurice Emery, Jyoti R. Patel, Annika Goos-Nilsson, Bryan K. Sorensen, Susan Swanson, David Arendsen, Gaoquan Li, James T. Link, Bach Nguyen
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:4169-4172
مصطلحات موضوعية: Nonsteroidal, Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, General Medicine, Metabolic stability, Pharmacology, Ligands, Biochemistry, chemistry.chemical_compound, Receptors, Glucocorticoid, Glucocorticoid receptor, Drug Discovery, medicine, Humans, Molecular Medicine, Molecular Biology, Glucocorticoid, Protein Binding, medicine.drug
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المؤلفون: Zhiqing He, Anthony J. Salerno, Harri Ahola, Paul Mak, Annika Goos-Nilsson
المصدر: Nucleic Acids Research. 24:566-572
مصطلحات موضوعية: Transcriptional Activation, Receptors, Retinoic Acid, Molecular Sequence Data, Retinoic acid, Saccharomyces cerevisiae, Biology, Retinoid X receptor, chemistry.chemical_compound, Transactivation, Genetics, Transcriptional regulation, Humans, Promoter Regions, Genetic, Transcription factor, Apolipoproteins A, Base Sequence, Retinoic Acid Receptor alpha, Gene Transfer Techniques, Molecular biology, body regions, Retinoic acid receptor, Retinoid X Receptors, chemistry, Nuclear receptor, Retinoic acid receptor alpha, embryonic structures, Research Article, Transcription Factors
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المؤلفون: Ronald C. Bernotas, Irene Feingold, James W. Jetter, Christofer Enroth, Anna Wilhelmsson, Robert W Morris, Christine Huselton, Annika Goos-Nilsson, John W. Ullrich, Jay E. Wrobel, Ponnal Nambi, Elaine Quinet, Rayomand J. Unwalla, Jeremy M. Travins
المصدر: Bioorganicmedicinal chemistry letters. 20(9)
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Sulfone, Cell Line, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Microsomes, Drug Discovery, medicine, Potency, Structure–activity relationship, Animals, Humans, Computer Simulation, Sulfones, Binding site, Liver X receptor, Molecular Biology, Binding selectivity, Liver X Receptors, Mice, Knockout, Binding Sites, Organic Chemistry, Quinoline, Atherosclerosis, Orphan Nuclear Receptors, Rats, Lipoproteins, LDL, chemistry, Quinolines, Molecular Medicine, lipids (amino acids, peptides, and proteins)
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المصدر: Analytical Biochemistry. 200:163-170
مصطلحات موضوعية: Steroid hormone receptor, Recombinant Fusion Proteins, medicine.medical_treatment, Biophysics, Endogeny, Ligands, medicine.disease_cause, Biochemistry, Gas Chromatography-Mass Spectrometry, Steroid, Pregnancy, Progesterone receptor, Escherichia coli, medicine, Humans, Receptor, Molecular Biology, Progesterone, Chemistry, DNA, Cell Biology, Chromatography, Ion Exchange, Ligand (biochemistry), Fusion protein, Female, Receptors, Progesterone
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المؤلفون: Jay E. Wrobel, Anna Wilhelmsson, Andrea Olland, Annika Goos-Nilsson, Elaine Quinet, Jeremy M. Travins, John W. Ullrich, Rayomand J. Unwalla, Robert R. Singhaus, Ponnal Nambi, Mark J. Evans, David H. Kaufman, Björn Kauppi, Ronald C. Bernotas
المصدر: Bioorganicmedicinal chemistry letters. 20(1)
مصطلحات موضوعية: Agonist, Hydrocarbons, Fluorinated, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, digestive system, Biochemistry, Sulfone, Cell Line, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Amide, Drug Discovery, polycyclic compounds, medicine, Potency, Animals, Humans, Computer Simulation, Sulfones, Liver X receptor, Molecular Biology, Liver X Receptors, Sulfonamides, Binding Sites, Aryl, Organic Chemistry, Quinoline, Hydrogen Bonding, Orphan Nuclear Receptors, Rats, chemistry, Nuclear receptor, Microsomes, Liver, Quinolines, Molecular Medicine, lipids (amino acids, peptides, and proteins), ATP-Binding Cassette Transporters, ATP Binding Cassette Transporter 1
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المؤلفون: Fletcher Horace, Elaine Quinet, John W. Ullrich, Mathias Färnegårdh, Annika Goos-Nilsson, Rayomand J. Unwalla, Ronald C. Bernotas, David H. Kaufman, Jay E. Wrobel, Anna Wilhelmsson, Ponnal Nambi, Robert R. Singhaus
المصدر: Bioorganicmedicinal chemistry. 17(4)
مصطلحات موضوعية: Agonist, Models, Molecular, Transcriptional Activation, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Receptors, Cytoplasmic and Nuclear, Crystallography, X-Ray, Ligands, Transfection, digestive system, Biochemistry, Cell Line, chemistry.chemical_compound, Mice, Amide, Drug Discovery, polycyclic compounds, medicine, Potency, Animals, Liver X receptor, Receptor, Molecular Biology, Liver X Receptors, biology, Organic Chemistry, food and beverages, Orphan Nuclear Receptors, Amides, DNA-Binding Proteins, Kinetics, chemistry, Gene Expression Regulation, Cell culture, ABCA1, biology.protein, Quinolines, Molecular Medicine, lipids (amino acids, peptides, and proteins), ATP-Binding Cassette Transporters, ATP Binding Cassette Transporter 1
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المؤلفون: Tomas Bonn, Michael Basso, Edward Martin Matelan, Shuguang Wang, Jay E. Wrobel, George P. Vlasuk, Christine Huselton, Anna Wilhelmsson, S. Marc Bowen, Robert John Steffan, Stephen J. Gardell, Elaine Quinet, Jason I. Reminick, Zamaratski Edouard, Annika Goos Nilsson, Tomas Hansson, Valerie Clerin, Mathias Färnegårdh, Rayomand J. Unwalla, Ronald L. Magolda, Ponnal Nambi, Mark J. Evans, Irene Feingold
المصدر: Journal of medicinal chemistry. 51(22)
مصطلحات موضوعية: Male, Models, Molecular, medicine.medical_specialty, Indazoles, Arteriosclerosis, Receptors, Cytoplasmic and Nuclear, Crystallography, X-Ray, Ligands, Partial agonist, Cell Line, Transactivation, Mice, Structure-Activity Relationship, Internal medicine, Cricetinae, Drug Discovery, medicine, Potency, Animals, Humans, Liver X receptor, Triglycerides, Liver X Receptors, Mice, Knockout, biology, Molecular Structure, Chemistry, Cell Differentiation, Hydrogen Bonding, Orphan Nuclear Receptors, Recombinant Proteins, DNA-Binding Proteins, Mice, Inbred C57BL, Fatty acid synthase, medicine.anatomical_structure, Endocrinology, Liver, Hepatocyte, ABCA1, LDL receptor, Models, Animal, biology.protein, Molecular Medicine, lipids (amino acids, peptides, and proteins)
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المؤلفون: Valerie Clerin, Robert R. Singhaus, Dawn A. Savio, Rayomand J. Unwalla, Elaine Quinet, Liang Chen, Baihua Hu, Annika Goos-Nilsson, Anita R Halpern, Christine Huselton, Irene Feingold, David H. Kaufman, Ronald C. Bernotas, Michael Basso, Qiang-Yuan Liu, Ponnal Nambi, Jay E. Wrobel, James W. Jetter, Farooq Azam, Anna Wilhelmsson, James C. Keith
المصدر: Bioorganicmedicinal chemistry. 15(10)
مصطلحات موضوعية: Agonist, Male, Transcriptional Activation, Spectrometry, Mass, Electrospray Ionization, Magnetic Resonance Spectroscopy, medicine.drug_class, Stereochemistry, Carboxylic acid, Clinical Biochemistry, Carboxylic Acids, Pharmaceutical Science, Receptors, Cytoplasmic and Nuclear, CHO Cells, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Apolipoproteins E, Cricetulus, In vivo, Cricetinae, Drug Discovery, medicine, Animals, Humans, Liver X receptor, Molecular Biology, Chromatography, High Pressure Liquid, Liver X Receptors, Phenylacetates, chemistry.chemical_classification, Mice, Knockout, Chemistry, Organic Chemistry, Quinoline, Aromatic amine, Atherosclerosis, Orphan Nuclear Receptors, Recombinant Proteins, DNA-Binding Proteins, Mice, Inbred C57BL, Nuclear receptor, Quinolines, Solvents, Molecular Medicine, lipids (amino acids, peptides, and proteins), Indicators and Reagents
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المؤلفون: Bradley J. Backes, Peer B. Jacobson, Phong Nguyen, Thomas W. von Geldern, Gregory Hamilton, Annika Goos-Nilsson, Steven Fung, Denise Wilcox, Marlena Grynfarb, Jiahong Wang
المصدر: Bioorganicmedicinal chemistry letters. 17(1)
مصطلحات موضوعية: Chemistry, Organic Chemistry, Clinical Biochemistry, Selection strategy, Pharmaceutical Science, Rats, Inbred Strains, Glucocorticoid Receptor Antagonists, Mifepristone, Pharmacology, Biochemistry, Rats, Receptors, Glucocorticoid, Pharmacokinetics, Liver, In vivo, Drug Discovery, medicine, Molecular Medicine, Animals, Molecular Biology, Glucocorticoids, medicine.drug