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1Academic Journal
المؤلفون: Michał Załuski, Tadeusz Karcz, Anna Drabczyńska, Christin Vielmuth, Agnieszka Olejarz-Maciej, Monika Głuch-Lutwin, Barbara Mordyl, Agata Siwek, Grzegorz Satała, Christa E. Müller, Katarzyna Kieć-Kononowicz
المصدر: Biomolecules, Vol 13, Iss 7, p 1079 (2023)
مصطلحات موضوعية: monoamine oxidase B inhibitors, adenosine A2A receptor antagonists, PDE4/10 inhibitors, D2 dopamine receptor agonists, Microbiology, QR1-502
وصف الملف: electronic resource
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2Academic Journal
المؤلفون: Magdalena Kotańska, Anna Dziubina, Małgorzata Szafarz, Kamil Mika, Karolina Reguła, Marek Bednarski, Małgorzata Zygmunt, Anna Drabczyńska, Jacek Sapa, Katarzyna Kieć-Kononowicz
المصدر: PLoS ONE, Vol 15, Iss 6, p e0229806 (2020)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/1932-6203
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3
المؤلفون: Clara T. Schoeder, Christa E. Müller, Andhika B Mahardhika, Katarzyna Kieć-Kononowicz, Anna Drabczyńska
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: Agonist, Orphan receptor, Cannabinoid receptor, 010405 organic chemistry, medicine.drug_class, Chemistry, medicine.medical_treatment, Organic Chemistry, Pharmacology, 01 natural sciences, Biochemistry, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, GPR55, Drug Discovery, medicine, GPR18, Cannabinoid, Receptor, G protein-coupled receptor
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4
المؤلفون: Christa E. Müller, Ewa Szymańska, Agata Doroz-Płonka, Tadeusz Karcz, Michał Załuski, Sonja Hinz, Jadwiga Handzlik, Katarzyna Kieć-Kononowicz, Jakub Schabikowski, Anna Drabczyńska, Katarzyna Stanuch, Gniewomir Latacz
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Molecular model, Stereochemistry, Organic Chemistry, Substituent, Pharmaceutical Science, Xanthine, Biochemistry, Adenosine receptor, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, chemistry, Docking (molecular), Amide, Drug Discovery, Molecular Medicine, Moiety, Acetamide
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5
المؤلفون: Jadwiga Handzlik, Christa E. Müller, Janina Karolak-Wojciechowska, Anna Drabczyńska, Katarzyna Kieć-Kononowicz, Andrzej Fruziński, Jakub Schabikowski, Agata Doroz-Płonka, Meryem Köse, Ewa Szymańska, Tadeusz Karcz
المصدر: Bioorganicmedicinal chemistry. 24(18)
مصطلحات موضوعية: 0301 basic medicine, Spectrophotometry, Infrared, Stereochemistry, Proton Magnetic Resonance Spectroscopy, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, Biochemistry, 03 medical and health sciences, Structure-Activity Relationship, Cricetulus, Drug Discovery, Structure–activity relationship, Animals, Humans, Homology modeling, Amino Acid Sequence, Binding site, Carbon-13 Magnetic Resonance Spectroscopy, Molecular Biology, chemistry.chemical_classification, Binding Sites, Sequence Homology, Amino Acid, Organic Chemistry, Antagonist, Receptors, Purinergic P1, Adenosine receptor, Affinities, Rats, 030104 developmental biology, chemistry, Docking (molecular), Xanthines, Molecular Medicine, Tricyclic
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6
المؤلفون: Anna, Dziubina, Karina, Szmyd, Małgorzata, Zygmunt, Jacek, Sapa, Magdalena, Dudek, Barbara, Filipek, Anna, Drabczyńska, Michał, Załuski, Karolina, Pytka, Katarzyna, Kieć-Kononowicz
المصدر: Pharmacological reports : PR. 68(6)
مصطلحات موضوعية: Male, Immobilization, Mice, Anti-Anxiety Agents, Dose-Response Relationship, Drug, Depression, Purinergic Agents, Drug Evaluation, Preclinical, Animals, Anxiety, Antidepressive Agents
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7
المؤلفون: Christa E. Müller, Jacek Sapa, Małgorzata Zygmunt, Katarzyna Kieć-Kononowicz, Barbara Filipek, Anna Drabczyńska
المصدر: Archiv der Pharmazie. 344:20-27
مصطلحات موضوعية: Male, Receptor, Adenosine A2A, Adenosine A2A Receptor Antagonists, Stereochemistry, Chemistry, Pharmaceutical Science, Adenosine A2A receptor, Reserpine, Pharmacology, Adenosine A2 Receptor Antagonists, Antiparkinson Agents, Mice, Pyrimidines, Parkinsonian Disorders, Adenosine a, Pharmacokinetics, Purines, Pyrazines, Drug Discovery, Oxotremorine, medicine, Animals, Potency, Receptor, medicine.drug
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8Predictive 3D-Quantitative Structure-Activity Relationship for A1 and A2A Adenosine Receptor Ligands
المؤلفون: Olga Yuzlenko, Anna Drabczyńska, Katarzyna Kieć-Kononowicz
المصدر: QSAR & Combinatorial Science. 28:1442-1454
مصطلحات موضوعية: Quantitative structure–activity relationship, Chemistry, Stereochemistry, Organic Chemistry, Substituent, Adenosine A2A receptor, Xanthine, Adenosine receptor, Computer Science Applications, chemistry.chemical_compound, Adenosine A1 receptor, Drug Discovery, Alkoxy group, Moiety
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9
المؤلفون: Karina Szmyd, Michał Załuski, Katarzyna Kieć-Kononowicz, Anna Drabczyńska, Jacek Sapa, Magdalena Dudek, Barbara Filipek, Karolina Pytka, Małgorzata Zygmunt, Anna Dziubina
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, medicine.medical_specialty, Chemistry, Adenosine A2A receptor, General Medicine, Antidepressant like, Anxiolytic like, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Endocrinology, Adenosine a, Animal models of depression, Internal medicine, medicine, 030217 neurology & neurosurgery
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10
المؤلفون: Andrzej Fruziński, Anke C. Schiedel, Olga Yuzlenko, Britta Schumacher, Weronika Zobnina, Christa E. Müller, Anna Drabczyńska, Janina Karolak-Wojciechowska, Katarzyna Kieć-Kononowicz
المصدر: Bioorganic & Medicinal Chemistry. 15:6956-6974
مصطلحات موضوعية: Male, Models, Molecular, Steric effects, Double bond, Stereochemistry, Clinical Biochemistry, Substituent, Pharmaceutical Science, Stereoisomerism, Crystallography, X-Ray, Ligands, Biochemistry, Chemical synthesis, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Animals, Structure–activity relationship, Computer Simulation, Molecular Biology, chemistry.chemical_classification, Binding Sites, Dose-Response Relationship, Drug, Molecular Structure, Receptor, Adenosine A1, Receptors, Adenosine A2, Chemistry, Organic Chemistry, Adenosine receptor, Disease Models, Animal, Models, Chemical, Purines, Lipophilicity, Molecular Medicine, Anticonvulsants, Injections, Intraperitoneal
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11
المؤلفون: Olga Yuzlenko, Anke C. Schiedel, Anna Drabczyńska, Katarzyna Kieć-Kononowicz, Britta Schumacher, Christa E. Müller, Janina Karolak-Wojciechowska
المصدر: Bioorganic & Medicinal Chemistry. 15:5003-5017
مصطلحات موضوعية: Models, Molecular, Magnetic Resonance Spectroscopy, Chemical Phenomena, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, Crystallography, X-Ray, Methylation, Biochemistry, Chemical synthesis, Propane, Structure-Activity Relationship, chemistry.chemical_compound, Adenosine A1 receptor, Cricetulus, Cricetinae, Drug Discovery, medicine, Animals, Receptor, Molecular Biology, Molecular Structure, Chemistry, Physical, Receptor, Adenosine A1, Receptors, Adenosine A2, Organic Chemistry, Benzene, Hydrogen Bonding, Xanthine, Ligand (biochemistry), Adenosine receptor, Adenosine, Rats, Pyrimidines, chemistry, Purines, Molecular Medicine, Pharmacophore, medicine.drug
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12
المؤلفون: Anna Drabczyńska, Elżbieta Pękala, Janina Karolak-Wojciechowska, Barbara Michalak, Katarzyna Kieć-Kononowicz, Britta Schumacher, Christa E. Müller
المصدر: European Journal of Medicinal Chemistry. 38:397-402
مصطلحات موضوعية: Receptor, Adenosine A2A, Stereochemistry, Substituent, adenosine receptors antagonists, Chemical synthesis, pyrimido[2,1-f]xanthines, Structure-Activity Relationship, chemistry.chemical_compound, Theophylline, adenosine A2A receptors antagonists, annelated xanthines, Drug Discovery, Animals, Humans, Receptor, Pharmacology, Molecular Structure, Chemistry, Aryl, Organic Chemistry, Receptors, Purinergic P1, Antagonist, Stereoisomerism, General Medicine, Xanthine, Adenosine receptor, Adenosine A2 Receptor Antagonists, Rats, Pyrimidines, Purinergic P1 Receptor Antagonists, Purines, Xanthines, Selectivity
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13
المؤلفون: Katarzyna Kieć-Kononowicz, Krystyna Gołembiowska, Anna Drabczyńska, Jacek Sapa, Małgorzata Zygmunt
مصطلحات موضوعية: Pharmacology, Antioxidant, medicine.drug_class, Adenosine A2A Receptor Antagonists, medicine.medical_treatment, Clinical Biochemistry, Catalepsy, Toxicology, medicine.disease, Biochemistry, Anti-inflammatory, Lipid peroxidation, Behavioral Neuroscience, chemistry.chemical_compound, chemistry, Adenosine a, medicine, Receptor, Antagonism, Biological Psychiatry
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14
المؤلفون: Małgorzata, Zygmunt, Krystyna, Gołembiowska, Anna, Drabczyńska, Katarzyna, Kieć-Kononowicz, Jacek, Sapa
المصدر: Pharmacology, biochemistry, and behavior. 132
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15
المؤلفون: Janina Karolak-Wojciechowska, H. Duddeck, Britta Schumacher, Christa E. Müller, S. Rockitt, Anna Drabczyńska, Barbara Michalak, Rudolf Wartchow, Elżbieta Pękala, Katarzyna Kieć-Kononowicz
المصدر: Pure and Applied Chemistry. 73:1411-1420
مصطلحات موضوعية: Chemistry, General Chemical Engineering, General Chemistry, Pharmacology, Purinergic signalling, Adenosine A3 receptor, Adenosine, Adenosine receptor, Metabotropic receptor, Dopamine receptor, medicine, Receptor, Adenosine A2B receptor, medicine.drug
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16
المؤلفون: Anna Drabczyńska, Rudolf Wartchow, Helmut Duddeck, Katarzyna Kieć-Kononowicz, Sven Rockitt
المصدر: Zeitschrift für Naturforschung B. 56:319-324
مصطلحات موضوعية: chemistry.chemical_compound, Trifluoromethyl, Phenylacetate, chemistry, Solid-state, Organic chemistry, General Chemistry, Xanthine, Medicinal chemistry
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17
المصدر: Scopus-Elsevier
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Stereochemistry, Organic Chemistry, Diastereomer, Molecule, Nuclear magnetic resonance spectroscopy, Physical and Theoretical Chemistry, Carbon-13 NMR, Methylene, Ring (chemistry), Chirality (chemistry), Chiral resolution
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::27e9bd9d191a708f08c44f5cb68b1121
https://doi.org/10.1002/1099-0690(200010)2000:20<3489::aid-ejoc3489>3.0.co;2-9 -
18
المؤلفون: M Gorczyca, D Malec, J Modzelewski, Maciej Pawłowski, Jacek Katlabi, Anna Drabczyńska
المصدر: European Journal of Medicinal Chemistry. 34:1085-1091
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Bicyclic molecule, medicine.drug_class, Stereochemistry, medicine.medical_treatment, Organic Chemistry, Analgesic, General Medicine, Chemical synthesis, chemistry.chemical_compound, Anticonvulsant, chemistry, Sedative, Drug Discovery, medicine, Lactam, Theophylline, Tricyclic, medicine.drug
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19
المؤلفون: Ewa Tatarczyńska, Anna Drabczyńska, Jacek Katlabi, Sijka Charakchieva-Minol, Maciej Pawłowski, Maria J. Mokrosz, A. Deren‐Wesolek, Ewa Chojnacka-Wójcik, Andrzej J. Bojarski, Beata Duszyńska
المصدر: European Journal of Medicinal Chemistry. 34:167-175
مصطلحات موضوعية: Pharmacology, Agonist, Purine, medicine.drug_class, Stereochemistry, Organic Chemistry, General Medicine, Chemical synthesis, Partial agonist, chemistry.chemical_compound, chemistry, Drug Discovery, medicine, Lactam, Receptor, Purine metabolism, 5-HT receptor
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20
المؤلفون: Pierre Koch, Christa E. Müller, Katarzyna Kieć-Kononowicz, Petra Küppers, Thomas Borrmann, Anna Drabczyńska, Rhalid Akkari, Meryem Köse, Miriam Schlenk, Andreas Brunschweiger, Jörg Hockemeyer, H. Radjainia
مصطلحات موضوعية: Purine, Drug, Monoamine Oxidase Inhibitors, Stereochemistry, media_common.quotation_subject, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, Adenosine A1 Receptor Antagonists, Biochemistry, chemistry.chemical_compound, Cricetulus, In vivo, Caffeine, Drug Discovery, medicine, Animals, Humans, Receptor, Molecular Biology, Monoamine Oxidase, media_common, Organic Chemistry, Neurodegeneration, Neurodegenerative Diseases, medicine.disease, Multiple target, Adenosine receptor, Adenosine A2 Receptor Antagonists, Monoamine neurotransmitter, chemistry, Purinergic P1 Receptor Antagonists, Purines, Xanthines, Molecular Medicine