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1
المؤلفون: Angelica E. Ehrenberg, Sofia Gustafsson, Muhammad Ikram Anwar, U. Helena Danielson, Gun Stenberg, Benjamin Schmuck
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry. 29:868-876
مصطلحات موضوعية: Cyclopropanes, Macrocyclic Compounds, Genotype, Lactams, Proline, Lactams, Macrocyclic, Hepatitis C virus, medicine.medical_treatment, Gene Expression, Hepacivirus, Isoindoles, Viral Nonstructural Proteins, Biology, medicine.disease_cause, Antiviral Agents, Genotype 1b, Drug Resistance, Viral, Drug Discovery, Escherichia coli, medicine, Protease Inhibitors, Cloning, Molecular, Pharmacology, chemistry.chemical_classification, Sulfonamides, NS3, Protease, Strain (chemistry), Genetic Variation, General Medicine, Hepatitis C, medicine.disease, Recombinant Proteins, Protein Structure, Tertiary, Thiazoles, Enzyme, Biochemistry, chemistry, Mutation, Quinolines, Carbamates, Oligopeptides
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2
المؤلفون: Eva Åkerblom, Robert Rönn, Angelica E. Ehrenberg, Anja Sandström, Göran Dahl, Pernilla Örtqvist, Anders Karlén, U. Helena Danielson, Aparna Vema
المصدر: Antiviral Therapy. 15:841-852
مصطلحات موضوعية: Models, Molecular, Pharmacology, Mutation rate, NS3, Protease, biology, medicine.medical_treatment, Hepatitis C virus, Hepacivirus, Drug resistance, Viral Nonstructural Proteins, biology.organism_classification, medicine.disease_cause, Virology, Structure-Activity Relationship, Flaviviridae, Infectious Diseases, Drug Resistance, Viral, medicine, Protease Inhibitors, Pharmacology (medical), Protease inhibitor (pharmacology), Pharmaceutical sciences, Protein Binding
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3
المؤلفون: Hiba Alogheli, Per Artursson, Anja Sandström, Richard Svensson, Eva Åkerblom, Angelica E. Ehrenberg, Anders Karlén, Anna Lampa, U. Helena Danielson
المصدر: Bioorganicmedicinal chemistry. 22(23)
مصطلحات موضوعية: Drug, Models, Molecular, Macrocyclic Compounds, Stereochemistry, media_common.quotation_subject, medicine.medical_treatment, Hepatitis C virus, Clinical Biochemistry, Substituent, Pharmaceutical Science, Drug resistance, Viral Nonstructural Proteins, Metathesis, medicine.disease_cause, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Humans, Protease Inhibitors, Molecular Biology, Cells, Cultured, media_common, NS3, Protease, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, Intracellular Signaling Peptides and Proteins, Dipeptides, In vitro, Pyrimidines, chemistry, Molecular Medicine, Caco-2 Cells, Carrier Proteins
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4
المؤلفون: Muhammad Ikram Anwar, Sofia Gustafsson, Angelica E. Ehrenberg, U. Helena Danielson, Benjamin Schmuck
المصدر: Journal of medicinal chemistry. 57(5)
مصطلحات موضوعية: chemistry.chemical_classification, NS3, Protease, viruses, medicine.medical_treatment, Hepatitis C virus, Kinetic analysis, Kinetics, virus diseases, Surface plasmon resonance biosensor, Biosensing Techniques, Surface Plasmon Resonance, Viral Nonstructural Proteins, medicine.disease_cause, Molecular biology, digestive system diseases, Enzyme, chemistry, Biochemistry, Drug Discovery, Genotype, medicine, Molecular Medicine, Protease Inhibitors
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5
المؤلفون: Mats Larhed, Angelica E. Ehrenberg, Eva Åkerblom, Anders Karlén, Richard Svensson, Anja Sandström, U. Helena Danielson, Hiba Alogheli, Per Artursson, Johan Gising, Anna Karin Belfrage
المصدر: Journal of medicinal chemistry. 57(5)
مصطلحات موضوعية: chemistry.chemical_classification, NS3, Protease, Binding Sites, Magnetic Resonance Spectroscopy, Molecular model, Peptidomimetic, Stereochemistry, medicine.medical_treatment, Stereoisomerism, Hepacivirus, Viral Nonstructural Proteins, Sulfonamide, chemistry, Biochemistry, Drug Discovery, Glycine, medicine, Molecular Medicine, Protease Inhibitors, Binding site
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6
المؤلفون: Anna Lampa, Aparna Vema, Eva Åkerblom, U. Helena Danielson, Anja Sandström, Anders Karlén, Angelica E. Ehrenberg, Gunnar Lindeberg
المصدر: Bioorganicmedicinal chemistry. 19(16)
مصطلحات موضوعية: Macrocyclic Compounds, Stereochemistry, Clinical Biochemistry, Glycine, Pharmaceutical Science, Hepacivirus, Viral Nonstructural Proteins, Metathesis, Virus Replication, Biochemistry, Antiviral Agents, Ring-closing metathesis, Cell Line, Tumor, Drug Discovery, Humans, Molecular Targeted Therapy, Enzyme Inhibitors, Microwaves, Molecular Biology, Inhibitory effect, Chemistry, Organic Chemistry, Hepatitis C, Chronic, Drug Design, Hcv ns3 protease, Molecular Medicine, Epimer, Linker, Cis–trans isomerism
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7
المؤلفون: Angelica E. Ehrenberg, Pernilla Örtqvist, Aparna Vema, Anders Karlén, Mats Larhed, U. Helena Danielson, Anneli Borg, Anja Sandström, Johan Gising
المصدر: Bioorganicmedicinal chemistry. 18(17)
مصطلحات موضوعية: Models, Molecular, Molecular model, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Substituent, Pharmaceutical Science, Tripeptide, Hepacivirus, Viral Nonstructural Proteins, Biochemistry, Chemical synthesis, Antiviral Agents, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Humans, Protease Inhibitors, Molecular Biology, NS3, Protease, Binding Sites, biology, Molecular Structure, Chemistry, Organic Chemistry, Enzyme inhibitor, Drug Design, Pyrazines, Glycine, biology.protein, Molecular Medicine, Protein Binding
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8
المؤلفون: Anna Lampa, Anders Karlén, Anja Sandström, Aparna Vema, Eva Åkerblom, U. Helena Danielson, Sofia Gustafsson, Angelica E. Ehrenberg, Gunnar Lindeberg
المصدر: Bioorganicmedicinal chemistry. 18(14)
مصطلحات موضوعية: Models, Molecular, Peptidomimetic, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Glycine, Pharmaceutical Science, Tripeptide, Hepacivirus, Viral Nonstructural Proteins, Biochemistry, Antiviral Agents, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Peptide synthesis, medicine, Structure–activity relationship, Humans, Protease Inhibitors, Molecular Biology, chemistry.chemical_classification, NS3, Protease, biology, Organic Chemistry, Hepatitis C, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine