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1Academic Journal
المصدر: International Symposium on the Chemistry of Natural Products. 1988, :232
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2Academic Journal
المؤلفون: Andrew T. McPhail, Donald R. McPhail, Kuo-Hsiung Lee, Masatake Niwa, Sheng-Teh Lu, Tian-Shung Wu, Yang-Chang Wu, Yoshimasa Hirata
المصدر: International Symposium on the Chemistry of Natural Products. 1988, :227
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3Academic Journal
المؤلفون: ANDREW T. MCPHAIL, BERNARD ROSENKRANTZ, DORIS SCHUMACHER, MOHINDAR S. PUAR, ROBERT S. JARET, TOM MOLLITOR
المصدر: The Journal of Antibiotics. 1992, 45(9):1540
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4Academic Journal
المؤلفون: ANDREW T. McPHAIL, KUO-HSIUNG LEE, LI-MING YANG, RONG-YANG Wu, TOSHIO YOKOI
المصدر: The Journal of Antibiotics. 1988, 41(4):488
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5Design, Synthesis, and X-ray Crystallographic Analysis of a Novel Class of HIV-1 Protease Inhibitors
المؤلفون: Andrew T. McPhail, Chih-Hung Wang, Christine Burlein, A. K. Ganguly, Yong Zhang, Steven S. Carroll, Corey Strickland, Dipshikha Biswas, Danielle Caroccia, Peter Orth, Vandna Munshi, S. Alluri, Eunhee Kang
المصدر: Journal of Medicinal Chemistry. 54:7176-7183
مصطلحات موضوعية: Models, Molecular, Protein Conformation, Thiazepines, Stereochemistry, medicine.medical_treatment, Crystallography, X-Ray, Radical cyclization, Structure-Activity Relationship, HIV Protease, HIV-1 protease, Drug Discovery, medicine, Protease, Molecular Structure, biology, Chemistry, Kazal-type serine protease inhibitor domain, Stereoisomerism, HIV Protease Inhibitors, Crystallography, Design synthesis, Drug Design, biology.protein, Molecular Medicine, Carbamates, Protein Binding
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6
المؤلفون: Hendrata Siska, Frank Bennett, Xiao Tong, Francisco Velazquez, Regina Huelgas, Kuo-Chi Cheng, Srikanth Venkatraman, Yuhua Huang, Andrew T. McPhail, Melissa Blackman, Patrick Pinto, Mousumi Sannigrahi, F. George Njoroge, Stephane L. Bogen, Raymond G. Lovey, Latha G. Nair, Ashok Arasappan
المصدر: Journal of Medicinal Chemistry. 53:3075-3085
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, Hepatitis C virus, Administration, Oral, Hepacivirus, Pharmacology, Crystallography, X-Ray, medicine.disease_cause, Sulfone, Structure-Activity Relationship, chemistry.chemical_compound, Pharmacokinetics, Oral administration, Boceprevir, Drug Discovery, medicine, Animals, Potency, Sulfones, Serine protease, biology, Ribavirin, Stereoisomerism, Haplorhini, Virology, digestive system diseases, Rats, chemistry, biology.protein, Molecular Medicine, Oligopeptides
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7
المؤلفون: Keith Eagen, Andrew T. McPhail, William J. Greenlee, Yunsheng Hsieh, Madhu Chintala, Samuel Chackalamannil, Yan Lin, Hsingan Tsai, Jayaram R. Tagat, Dario Doller, Ho-Sam Ahn, Yan Xia, George Boykow, Martin C. Clasby, Jacqueline Agans-Fantuzzi, Michael Czarniecki
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:3647-3651
مصطلحات موضوعية: Platelet Aggregation, Chemistry, Pharmaceutical, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Naphthalenes, Ligands, Biochemistry, Inhibitory Concentration 50, chemistry.chemical_compound, Alkaloids, Thrombin, Piperidines, In vivo, Drug Discovery, Thrombin receptor, medicine, Animals, Furans, Molecular Biology, IC50, chemistry.chemical_classification, Chemistry, Organic Chemistry, Parasympatholytics, Biological activity, In vitro, Rats, Macaca fascicularis, Models, Chemical, Area Under Curve, Himbacine, Molecular Medicine, Receptors, Thrombin, Protein Binding, medicine.drug, Tricyclic
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8
المؤلفون: Lynn A. Hyde, John W. Clader, Eric M. Parker, Zhiqiang Zhao, Lili Zhang, Andrew T. McPhail, Lixin Song, Amin A. Nomeir, Gwendolyn T. Wong, Wei Li, William J. Greenlee, Qi Zhang, Hubert B. Josien, Murali Rajagopalan, Dmitri A. Pissarnitski, Thomas A. Bara, Theodros Asberom
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:511-516
مصطلحات موضوعية: Models, Molecular, Magnetic Resonance Spectroscopy, Transgene, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Mice, Transgenic, Pharmacology, Crystallography, X-Ray, Biochemistry, Amyloid beta-Protein Precursor, Mice, Structure-Activity Relationship, Alzheimer Disease, In vivo, Drug Discovery, medicine, Amyloid precursor protein, Animals, Humans, Structure–activity relationship, Potency, Enzyme Inhibitors, Molecular Biology, Amyloid beta-Peptides, biology, Chemistry, Organic Chemistry, medicine.disease, Rats, Enzyme inhibitor, Area Under Curve, biology.protein, Molecular Medicine, Indicators and Reagents, Amyloid Precursor Protein Secretases, Alzheimer's disease, Amyloid precursor protein secretase
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9
المؤلفون: Hendrata Siska, Rebecca Osterman, Andrew T. McPhail, Yuhua Huang, Patrick Pinto, C. Anderson Evans, Frank Bennett, Tze-Ming Chan, Mousumi Sannigrahi, Alexei V. Buevich
المصدر: Tetrahedron Letters. 47:6469-6472
مصطلحات موضوعية: chemistry.chemical_classification, Hexane, chemistry.chemical_compound, Chemistry, Carboxylic acid, Organic Chemistry, Drug Discovery, Organic chemistry, Biochemistry, Cyclopropane
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10
المؤلفون: George Boykow, Samuel Chackalamannil, Andrew T. McPhail, Hsingan Tsai, William J. Greenlee, Yan Xia, Dario Doller, Ho-Sam Ahn, Michael Czarniecki, Yuguang Wang, Tze-Ming Chan, Keith Eagen
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:4969-4972
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Naphthalenes, Ring (chemistry), Biochemistry, Inhibitory Concentration 50, Lactones, Structure-Activity Relationship, chemistry.chemical_compound, Alkaloids, Piperidines, Drug Discovery, Thrombin receptor, Pyridine, Structure–activity relationship, Receptor, PAR-1, Furans, Molecular Biology, chemistry.chemical_classification, Molecular Structure, Chemistry, Organic Chemistry, Himbacine, Michael reaction, Molecular Medicine, Stereoselectivity, Lactone
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11
المؤلفون: Mahesh J. Patel, † Tze-Ming Chan, Bahige Baroudy, Joseph Terracciano, Mohindar S. Puar, Min Chu, Nicole Wagner, Vincent P. Gullo, and Andrew T. McPhail, Ronald Mierzwa, † Shu-Wei Yang
المصدر: Journal of Natural Products. 69:1025-1028
مصطلحات موضوعية: Spectrometry, Mass, Electrospray Ionization, Anti-HIV Agents, Stereochemistry, Pharmaceutical Science, Chaetomium, Pharmacognosy, Crystallography, X-Ray, Heterocyclic Compounds, 4 or More Rings, Analytical Chemistry, Inhibitory Concentration 50, Chemokine receptor, Drug Discovery, Humans, Receptor, IC50, Pharmacology, Molecular Structure, Chaetomium globosum, Chemistry, Organic Chemistry, Arizona, Biological activity, In vitro, Plant Leaves, Complementary and alternative medicine, Biochemistry, CCR5 Receptor Antagonists, Molecular Medicine, Two-dimensional nuclear magnetic resonance spectroscopy
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12
المؤلفون: Andrew T. McPhail, Dong Xiao, Neng-Yang Shih, Brian J. Lavey, Anandan Palani, Gerard P. Randolph, Robert G. Aslanian, Jean E. Lachowicz, Joseph A. Kozlowski, Cheng Wang, Ruth A. Duffy
المصدر: Tetrahedron Letters. 46:7653-7656
مصطلحات موضوعية: 2-phenylpiperidine, chemistry.chemical_compound, chemistry, Ligand, Stereochemistry, Organic Chemistry, Drug Discovery, Electrophile, NK1 receptor antagonist, Piperidine, Biochemistry, Pyrrolidine, Carbanion
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13
المؤلفون: Tze-Ming Chan, J. Misiaszek, C.H. Wang, Andrew T. McPhail, A.K. Ganguly, Birendra N. Pramanik
المصدر: Tetrahedron Letters. 45:8909-8912
مصطلحات موضوعية: Chemistry, Radical, Organic Chemistry, Drug Discovery, Photochemistry, Biochemistry, Radical cyclization, Mechanism (sociology)
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14
المؤلفون: Gordon M. Cragg, Kenneth F. Bastow, Fang Rong Chang, Kuo Hsiung Lee, Andrew T. McPhail, Ken-ichiro Hayashi, Yuka Nakanishi, Hiroshi Nozaki
المصدر: Journal of Natural Products. 67:990-993
مصطلحات موضوعية: Stereochemistry, Lantana, Pharmaceutical Science, Analytical Chemistry, Inhibitory Concentration 50, Drug Discovery, Tumor Cells, Cultured, Ic50 values, Humans, Cytotoxic T cell, Nuclear Magnetic Resonance, Biomolecular, Pharmacology, Plants, Medicinal, Molecular Structure, biology, Chemistry, Puerto Rico, Organic Chemistry, biology.organism_classification, Antineoplastic Agents, Phytogenic, Human tumor, Complementary and alternative medicine, Drug Resistance, Neoplasm, Cell culture, Molecular Medicine, Lantana involucrata, Drug Screening Assays, Antitumor, Naphthoquinones
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15
المؤلفون: Anil K. Saksena, Andrew T. McPhail, Tze-Ming Chan, Pradip R. Das, Ashit K. Ganguly, Rebecca Osterman, Birendra N. Pramanik, Viyyoor M. Girijavallabhan, Mccormick Jinping
المصدر: Tetrahedron Letters. 44:7997-8000
مصطلحات موضوعية: chemistry.chemical_compound, Olefin fiber, chemistry, Stereochemistry, Aryl, Organic Chemistry, Drug Discovery, Substituent, chemistry.chemical_element, Stereoselectivity, Biochemistry, Nitrogen
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16
المؤلفون: Viyyoor M. Girijavallabhan, Andrew T. McPhail, Pradip R. Das, Anil K. Saksena, Birendra N. Pramanik, Mohindar S. Puar
المصدر: Tetrahedron Letters. 44:7201-7204
مصطلحات موضوعية: Stereochemistry, Mesylate, Organic Chemistry, Alcohol, Uracil, General Medicine, Biochemistry, Medicinal chemistry, Acetonide, chemistry.chemical_compound, chemistry, Group (periodic table), Product (mathematics), Drug Discovery, Mitsunobu reaction, Single crystal
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17
المؤلفون: Neng-Yang Shih, Andrew T. McPhail, Ho-Jane Shue, Xiao Chen, David J. Blythin, John C. Anthes, Piwinski John J
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:3161-3165
مصطلحات موضوعية: Male, Models, Molecular, medicine.drug_class, Stereochemistry, Guinea Pigs, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Carboxamide, In Vitro Techniques, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Piperazines, Structure-Activity Relationship, chemistry.chemical_compound, Vas Deferens, Piperidines, Cricetinae, Drug Discovery, medicine, Animals, Structure–activity relationship, Amino Acids, Derivatization, Receptor, Molecular Biology, Organic Chemistry, Dual inhibitor, Stereoisomerism, Receptors, Neurokinin-2, General Medicine, Receptors, Neurokinin-1, Trachea, Piperazine, Chromatographic separation, chemistry, Molecular Medicine, Enantiomer, Derivative (chemistry)
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18
المؤلفون: Tong Gan, Andrew T. McPhail, George S. K. Wong, Spitler James M, Ingrid Mergelsberg, Ramani R. Raghavan, John K. Jenkins, Alan J. Miller, Gregory A. Reichard
المصدر: Tetrahedron: Asymmetry. 13:939-943
مصطلحات موضوعية: Inorganic Chemistry, chemistry.chemical_compound, Core fragment, chemistry, Stereochemistry, Organic Chemistry, Michael reaction, Enantioselective synthesis, Physical and Theoretical Chemistry, Catalysis, Acetamide
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19
المصدر: The Journal of Organic Chemistry. 67:3152-3155
مصطلحات موضوعية: chemistry.chemical_classification, Depsipeptide, Stereochemistry, Carboxylic acid, Organic Chemistry, chemistry.chemical_element, Esters, Ether, Crystallography, X-Ray, Peptides, Cyclic, Combinatorial chemistry, Chemical synthesis, Catalysis, Ruthenium, chemistry.chemical_compound, chemistry, Cyclization, Yield (chemistry), Combinatorial Chemistry Techniques, Chromatography, Thin Layer, Phenols, Nuclear Magnetic Resonance, Biomolecular, Ethers
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20
المؤلفون: Mohamed S. Ahmed, Farouk S. El-Feraly, Ahmed M. Galal, Mahmoud A. ElSohly, Andrew T. McPhail, Hala N. ElSohly, Samir A. Ross
المصدر: Journal of Natural Products. 65:184-188
مصطلحات موضوعية: Lung Neoplasms, Magnetic Resonance Spectroscopy, Photochemistry, Dimer, Molecular Conformation, Saudi Arabia, Pharmaceutical Science, Breast Neoplasms, Ether, Crystallography, X-Ray, Chemical synthesis, Analytical Chemistry, Structure-Activity Relationship, chemistry.chemical_compound, Carcinoma, Non-Small-Cell Lung, Drug Discovery, Pyridine, Tumor Cells, Cultured, Humans, Organic chemistry, Triphenylphosphine, Pharmacology, Molecular Structure, Organic Chemistry, Stereoisomerism, Antineoplastic Agents, Phytogenic, Artemisinins, Oxygen, Acetic anhydride, Artemisia, Complementary and alternative medicine, chemistry, Molecular Medicine, Hemiacetal, Photooxygenation, Female, Drug Screening Assays, Antitumor, Oxidation-Reduction, Sesquiterpenes