المؤلفون: Haidar, Samer, Amesty, Ángel, Oramas-Royo, Sandra, Götz, Claudia, El-Awaad, Ehab, Kaiser, Jana, Bödecker, Sarah, Arnold, Amelie, Aichele, Dagmar, Amaro-Luis, Juan M., Estévez-Braun, Ana, Jose, Joachim

المصدر: Bioorganic & Medicinal Chemistry ; volume 105, page 117727 ; ISSN 0968-0896

الاتاحة: http://dx.doi.org/10.1016/j.bmc.2024.117727
https://api.elsevier.com/content/article/PII:S096808962400141X?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S096808962400141X?httpAccept=text/plain

المؤلفون: Aichele, Dagmar

Relation: https://doi.org/10.5281/zenodo.12788457; https://doi.org/10.5281/zenodo.12788458; oai:zenodo.org:12788458

الاتاحة: https://doi.org/10.5281/zenodo.12788458

المؤلفون: Rumler, Hendrik, Schmithals, Claudia, Werner, Christian, Bollacke, Andre, Aichele, Dagmar, Götz, Claudia, Niefind, Karsten, Wünsch, Bernhard, Jose, Joachim

المصدر: ACS Pharmacology & Translational Science; 12/13/2024, Vol. 7 Issue 12, p3846-3866, 21p

المؤلفون: López-Rojas, Priscila, Haidar, Samer, Jürgens, Franziska M., Aichele, Dagmar, Amesty, Ángel, Estévez-Braun, Ana, Jose, Joachim

المصدر: Results in Chemistry ; volume 6, page 100997 ; ISSN 2211-7156

الاتاحة: http://dx.doi.org/10.1016/j.rechem.2023.100997
https://api.elsevier.com/content/article/PII:S2211715623002369?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S2211715623002369?httpAccept=text/plain

المؤلفون: Birus, Robin, El‐awaad, Ehab, Ballentin, Laurens, Alchab, Faten, Aichele, Dagmar, Ettouati, Laurent, Götz, Claudia, Le Borgne, Marc, Jose, Joachim

المساهمون: Westfälische Wilhelms-Universität Münster = University of Münster (WWU), Assiut University, Molécules bioactives et chimie médicinale (B2MC), Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon, Manara University, Institut de Chimie et Biochimie Moléculaires et Supramoléculaires (ICBMS), Université de Lyon-Université de Lyon-École Supérieure de Chimie Physique Électronique de Lyon (CPE)-Institut National des Sciences Appliquées de Lyon (INSA Lyon), Université de Lyon-Institut National des Sciences Appliquées (INSA)-Institut National des Sciences Appliquées (INSA)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS), Universität des Saarlandes Saarbrücken = Saarland University Saarbrücken, Centre de Recherche en Cancérologie de Lyon (UNICANCER/CRCL), Centre Léon Bérard Lyon -Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS), Centre Léon Bérard Lyon

المصدر: ISSN: 2211-5463.

مصطلحات موضوعية: CK2, HPLC-MS/MS, indeno[1, 2-b]indole, live cell imaging, pharmacokinetics, [SDV.SP.PHARMA]Life Sciences [q-bio]/Pharmaceutical sciences/Pharmacology, [SDV.CAN]Life Sciences [q-bio]/Cancer

Relation: info:eu-repo/semantics/altIdentifier/pmid/34873879; PUBMED: 34873879; PUBMEDCENTRAL: PMC8804612

الاتاحة: https://hal.science/hal-03471998
https://hal.science/hal-03471998v1/document
https://hal.science/hal-03471998v1/file/10.1002_2211-5463.13346.pdf
https://doi.org/10.1002/2211-5463.13346

المؤلفون: Rumler, Hendrik, Schmithals, Claudia, Werner, Christian, Bollacke, Andre, Aichele, Dagmar, Götz, Claudia, Niefind, Karsten, Wünsch, Bernhard, Jose, Joachim

المصدر: ACS Pharmacol Transl Sci ; ISSN:2575-9108 ; Volume:7 ; Issue:12

Relation: https://doi.org/10.1021/acsptsci.4c00426; https://pubmed.ncbi.nlm.nih.gov/39698287; https://www.ncbi.nlm.nih.gov/pmc/articles/PMC11651316/

الاتاحة: https://doi.org/10.1021/acsptsci.4c00426
https://pubmed.ncbi.nlm.nih.gov/39698287
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC11651316/

المؤلفون: El-Awaad, Ehab, Birus, Robin, Marminon, Christelle, Bouaziz, Zouhair, Ballentin, Laurens, Aichele, Dagmar, Le Borgne, Marc, Jose, Joachim

المساهمون: Westfälische Wilhelms-Universität Münster = University of Münster (WWU), Centre de Recherche en Cancérologie de Lyon (UNICANCER/CRCL), Centre Léon Bérard Lyon -Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS), Molécules bioactives et chimie médicinale (B2MC), Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon

المصدر: ISSN: 1424-8247 ; Pharmaceuticals ; https://hal.science/hal-03311530 ; Pharmaceuticals, 2021, 14 (6), pp.542. ⟨10.3390/ph14060542⟩.

مصطلحات موضوعية: CK2 inhibitor, LC-MS, anticancer, indeno[1 2-b]indole, pharmacokinetics, [SDV.SP.PHARMA]Life Sciences [q-bio]/Pharmaceutical sciences/Pharmacology, [CHIM.THER]Chemical Sciences/Medicinal Chemistry, [SDV.CAN]Life Sciences [q-bio]/Cancer

Relation: info:eu-repo/semantics/altIdentifier/pmid/34198928; hal-03311530; https://hal.science/hal-03311530; https://hal.science/hal-03311530/document; https://hal.science/hal-03311530/file/pharmaceuticals-14-00542-v2.pdf; PUBMED: 34198928

الاتاحة: https://hal.science/hal-03311530
https://hal.science/hal-03311530/document
https://hal.science/hal-03311530/file/pharmaceuticals-14-00542-v2.pdf
https://doi.org/10.3390/ph14060542

المؤلفون: Haidar, Samer, Marminon, Christelle, Aichele, Dagmar, Nacereddine, Abdelhamid, Zeinyeh, Wael, Bouzina, Abdeslem, Berredjem, Malika, Ettouati, Laurent, Bouaziz, Zouhair, Le Borgne, Marc, Jose, Joachim

المساهمون: Westfälische Wilhelms-Universität Münster = University of Münster (WWU), Molécules bioactives et chimie médicinale (B2MC), Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon, Université Badji Mokhtar Annaba (UBMA)

المصدر: ISSN: 1420-3049 ; Molecules ; https://hal.science/hal-02424862 ; Molecules, 2020, 25 (1), pp.97. ⟨10.3390/molecules25010097⟩ ; https://www.mdpi.com/1420-3049/25/1/97.

مصطلحات موضوعية: 3-b]furan-4, 9-dione, indeno[1, 2-b]indole, cancer, naphtho[2, CK2, QSAR, [SDV.SP.PHARMA]Life Sciences [q-bio]/Pharmaceutical sciences/Pharmacology, [SDV.SP.MED]Life Sciences [q-bio]/Pharmaceutical sciences/Medication, [CHIM.THER]Chemical Sciences/Medicinal Chemistry, [CHIM.CHEM]Chemical Sciences/Cheminformatics

Relation: hal-02424862; https://hal.science/hal-02424862; https://hal.science/hal-02424862/document; https://hal.science/hal-02424862/file/molecules-25-00097.pdf

الاتاحة: https://hal.science/hal-02424862
https://hal.science/hal-02424862/document
https://hal.science/hal-02424862/file/molecules-25-00097.pdf
https://doi.org/10.3390/molecules25010097

المؤلفون: Estévez Braun, Ana María, Oramas-Royo, Sandra M., Haidar, Samer, Amesty Arrieta, Ángel Ernesto, Martín-Acosta, Pedro, Feresin, Gabriela, Tapia, Alejandro, Aichele, Dagmar, Jose, Joachim

وصف الملف: application/pdf

Relation: http://riull.ull.es/xmlui/handle/915/18632

الاتاحة: http://riull.ull.es/xmlui/handle/915/18632

المؤلفون: Birus, Robin, El-Awaad, Ehab, Ballentin, Laurens, Alchab, Faten, Aichele, Dagmar, Ettouati, Laurent, Götz, Claudia, Le Borgne, Marc, Jose, Joachim

المساهمون: Universitäts- und Landesbibliothek Münster, Westfälische Wilhelms-Universität Münster = University of Münster (WWU), Assiut University, Molécules bioactives et chimie médicinale (B2MC), Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon, Santé Lyon Est - Louis Léopold Ollier, Université de Lyon-Université de Lyon-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS), Institut de Chimie et Biochimie Moléculaires et Supramoléculaires (ICBMS), Université de Lyon-Université de Lyon-École Supérieure de Chimie Physique Électronique de Lyon (CPE)-Institut National des Sciences Appliquées de Lyon (INSA Lyon), Université de Lyon-Institut National des Sciences Appliquées (INSA)-Institut National des Sciences Appliquées (INSA)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS), Saarland University [Saarbrücken], Centre de Recherche en Cancérologie de Lyon (UNICANCER/CRCL), Centre Léon Bérard [Lyon]-Université Claude Bernard Lyon 1 (UCBL), Centre Léon Bérard [Lyon], Le Borgne, Marc, Westfälische Wilhelms-Universität Münster (WWU), Université de Lyon-Université de Lyon-Institut National des Sciences Appliquées de Lyon (INSA Lyon), Université de Lyon-Institut National des Sciences Appliquées (INSA)-Institut National des Sciences Appliquées (INSA)-Institut de Chimie du CNRS (INC)-École Supérieure Chimie Physique Électronique de Lyon-Centre National de la Recherche Scientifique (CNRS)

المصدر: FEBS Open Bio
FEBS Open Bio, 2022, 12, pp.394-411. ⟨10.1002/2211-5463.13346⟩
FEBS Open Bio, Wiley Open Access/Elsevier, 2021, ⟨10.1002/2211-5463.13346⟩
FEBS Open Bio, Vol 12, Iss 2, Pp 394-411 (2022)

مصطلحات موضوعية: 540 Chemistry and allied sciences, Indoles, HPLC‐MS/MS, [SDV.SP.MED] Life Sciences [q-bio]/Pharmaceutical sciences/Medication, QH301-705.5, CK2, [CHIM.THER] Chemical Sciences/Medicinal Chemistry, indeno[1, [CHIM.THER]Chemical Sciences/Medicinal Chemistry, [SDV.SP.MED]Life Sciences [q-bio]/Pharmaceutical sciences/Medication, Naphthyridines, Biology (General), Casein Kinase II, Research Articles, live‐cell imaging, HPLC-MS/MS, indeno[1,2‐b]indole, Chemistry and allied sciences, live cell imaging, 2-b]indole, [SDV.SP.PHARMA] Life Sciences [q-bio]/Pharmaceutical sciences/Pharmacology, ddc:540, indeno[1,2-b]indole, live-cell imaging, pharmacokinetics, [SDV.SP.PHARMA]Life Sciences [q-bio]/Pharmaceutical sciences/Pharmacology, Phenazines, Research Article

وصف الملف: application/pdf

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aa5fc80887648f7dbe36bac662669c89
https://repositorium.uni-muenster.de/transfer/miami/e07de578-a357-4ad5-a2a9-5e6e1e7da84e

المؤلفون: Hochscherf, Jennifer, Lindenblatt, Dirk, Witulski, Benedict, Birus, Robin, Aichele, Dagmar, Marminon, Christelle, Bouaziz, Zouhair, Le Borgne, Marc, Jose, Joachim, Niefind, Karsten

المساهمون: Westfälische Wilhelms-Universität Münster = University of Münster (WWU), Molécules bioactives et chimie médicinale (B2MC), Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon

المصدر: ISSN: 1424-8247 ; Pharmaceuticals ; https://hal.science/hal-01683237 ; Pharmaceuticals, 2017, 10 ((4)98), ⟨10.3390/ph10040098⟩.

مصطلحات موضوعية: ATP-competitive inhibitors, 2-b]indole scaffold, membrane permeability, indeno[1, paralogous isoforms CK2α and CK2α, dual inhibitors, protein kinase CK2, casein kinase 2, [CHIM.THER]Chemical Sciences/Medicinal Chemistry, [CHIM.CRIS]Chemical Sciences/Cristallography, [SDV.CAN]Life Sciences [q-bio]/Cancer, [SDV.SP]Life Sciences [q-bio]/Pharmaceutical sciences, [SDV.BBM.BS]Life Sciences [q-bio]/Biochemistry, Molecular Biology/Structural Biology [q-bio.BM]

Relation: info:eu-repo/semantics/altIdentifier/pmid/29236079; hal-01683237; https://hal.science/hal-01683237; https://hal.science/hal-01683237/document; https://hal.science/hal-01683237/file/pharmaceuticals-10-00098-v4-MLB.pdf; PUBMED: 29236079; PUBMEDCENTRAL: PMC5748653

الاتاحة: https://hal.science/hal-01683237
https://hal.science/hal-01683237/document
https://hal.science/hal-01683237/file/pharmaceuticals-10-00098-v4-MLB.pdf
https://doi.org/10.3390/ph10040098

المؤلفون: Birus, Robin, El-Awaad, Ehab, Ballentin, Laurens, Alchab, Faten, Aichele, Dagmar, Ettouati, Laurent, Götz, Claudia, Le Borgne, Marc, Jose, Joachim

المساهمون: Westfälische Wilhelms-Universität Münster = University of Münster (WWU), Molécules bioactives et chimie médicinale (B2MC), Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon, Centre de Recherche en Cancérologie de Lyon (UNICANCER/CRCL), Centre Léon Bérard Lyon -Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS)

المصدر: 7th International Electronic Conference on Medicinal Chemistry
https://hal.science/hal-03552581
7th International Electronic Conference on Medicinal Chemistry, Nov 2021, Basel, Switzerland. pp.11450, ⟨10.3390/ECMC2021-11450⟩
https://ecmc2022.sciforum.net/

مصطلحات موضوعية: Anti-cancer, CK2, Indeno[1, 2-b]indole, Live cell imaging, Subcellular distribution, [SDV.SP.PHARMA]Life Sciences [q-bio]/Pharmaceutical sciences/Pharmacology, [SDV.SP.MED]Life Sciences [q-bio]/Pharmaceutical sciences/Medication, [CHIM.THER]Chemical Sciences/Medicinal Chemistry

جغرافية الموضوع: Basel, Switzerland

Relation: hal-03552581; https://hal.science/hal-03552581

الاتاحة: https://hal.science/hal-03552581
https://doi.org/10.3390/ECMC2021-11450

المؤلفون: Birus, Robin, Marminon, Christelle, Aichele, Dagmar, Haidar, Samer, Ousset, Marine, Ettouati, Laurent, Alchab, Faten, Audebert, Solène, Rolland de Ravel, Marc, Pinaud, Noël, Bouaziz, Zouhair, Guillon, Jean, Jose, Joachim, Le Borgne, Marc

المساهمون: Westfälische Wilhelms-Universität Münster = University of Münster (WWU), Centre de Recherche en Cancérologie de Lyon (UNICANCER/CRCL), Centre Léon Bérard Lyon -Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS), Molécules bioactives et chimie médicinale (B2MC), Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon

المصدر: 6th International Electronic Conference on Medicinal Chemistry
https://hal.science/hal-03566434
6th International Electronic Conference on Medicinal Chemistry, Nov 2020, Basel, Switzerland. pp.7433, ⟨10.3390/ECMC2020-07433⟩
https://ecmc2020.sciforum.net/

مصطلحات موضوعية: [SDV.SP.PHARMA]Life Sciences [q-bio]/Pharmaceutical sciences/Pharmacology, [SDV.SP.MED]Life Sciences [q-bio]/Pharmaceutical sciences/Medication, [CHIM.THER]Chemical Sciences/Medicinal Chemistry

جغرافية الموضوع: Basel, Switzerland

Relation: hal-03566434; https://hal.science/hal-03566434

الاتاحة: https://hal.science/hal-03566434
https://doi.org/10.3390/ECMC2020-07433

المؤلفون: Haidar, Samer, Jürgens, Franziska, Aichele, Dagmar, Jose, Joachim

المصدر: Current Computer-Aided Drug Design ; volume 17, issue 2, page 323-331 ; ISSN 1573-4099

الاتاحة: http://dx.doi.org/10.2174/1573409916666200311150744
https://www.eurekaselect.com/article/download/180116
https://www.eurekaselect.com/180116/article

المؤلفون: Oramas-Royo, Sandra, Haidar, Samer, Amesty, Ángel, Martín-Acosta, Pedro, Feresin, Gabriela, Tapia, Alejandro, Aichele, Dagmar, Jose, Joachim, Estévez-Braun, Ana

المساهمون: Spanish MINECO SAF, MICINN, Gobierno Autónomo Canario, European Regional Development Fund, Cabildo de Tenerife, PMA

المصدر: Bioorganic Chemistry ; volume 95, page 103520 ; ISSN 0045-2068

الاتاحة: http://dx.doi.org/10.1016/j.bioorg.2019.103520
https://api.elsevier.com/content/article/PII:S0045206819316566?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S0045206819316566?httpAccept=text/plain

المؤلفون: Birus, Robin, El‐Awaad, Ehab, Ballentin, Laurens, Alchab, Faten, Aichele, Dagmar, Ettouati, Laurent, Götz, Claudia, Le Borgne, Marc, Jose, Joachim

المصدر: FEBS Open Bio; Feb2022, Vol. 12 Issue 2, p394-411, 18p

مصطلحات موضوعية: PROTEIN kinase CK2, INDOLE, CELL migration, CELL analysis, CANCER cells, INDOLE derivatives

المؤلفون: Martín-Acosta, Pedro, Haider, Samer, Amesty, Ángel, Aichele, Dagmar, Jose, Joachim, Estévez-Braun, Ana

المساهمون: Spanish MINECO SAF, European Regional Development Fund (FEDER)

المصدر: European Journal of Medicinal Chemistry ; volume 144, page 410-423 ; ISSN 0223-5234

الاتاحة: http://dx.doi.org/10.1016/j.ejmech.2017.12.058
https://api.elsevier.com/content/article/PII:S0223523417310899?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S0223523417310899?httpAccept=text/plain

المؤلفون: Aichele, Dagmar, Le Borgne, Marc, Jose, Joachim

المساهمون: Westfälische Wilhelms-Universität Münster = University of Münster (WWU), Molécules bioactives et chimie médicinale (B2MC), Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon

المصدر: Pharmaceuticals ; Second International Electronic Conference on Medicinal Chemistry (ECMC-2) ; https://hal.science/hal-01683452 ; Second International Electronic Conference on Medicinal Chemistry (ECMC-2), Nov 2016, Bâle, Switzerland. pp.15/A021, ⟨10.3390/ph10010020⟩

مصطلحات موضوعية: drug discovery, biomolecules, biological and therapeutic targets, medicinal chemistry, pharmacological evaluation, drug development, [CHIM.THER]Chemical Sciences/Medicinal Chemistry, [SDV.BBM]Life Sciences [q-bio]/Biochemistry, Molecular Biology, [SDV.CAN]Life Sciences [q-bio]/Cancer, [SDV.SP]Life Sciences [q-bio]/Pharmaceutical sciences

جغرافية الموضوع: Bâle, Switzerland

Relation: info:eu-repo/semantics/altIdentifier/pmid/28146112; hal-01683452; https://hal.science/hal-01683452; PUBMED: 28146112; PUBMEDCENTRAL: PMC5374424

الاتاحة: https://hal.science/hal-01683452
https://doi.org/10.3390/ph10010020

المؤلفون: Hochscherf, Jennifer, Lindenblatt, Dirk, Witulski, Benedict, Birus, Robin, Aichele, Dagmar, Marminon, Christelle, Bouaziz, Zouhair, Le Borgne, Marc, Jose, Joachim, Niefind, Karsten

مصطلحات موضوعية: ddc:no

Relation: Hochscherf, Jennifer orcid:0000-0002-4412-7391 , Lindenblatt, Dirk, Witulski, Benedict, Birus, Robin, Aichele, Dagmar, Marminon, Christelle orcid:0000-0002-4043-3949 , Bouaziz, Zouhair, Le Borgne, Marc orcid:0000-0003-1398-075X , Jose, Joachim and Niefind, Karsten orcid:0000-0002-0183-6315 (2017). Unexpected Binding Mode of a Potent Indeno[1,2-b]indole-Type Inhibitor of Protein Kinase CK2 Revealed by Complex Structures with the Catalytic Subunit CK2 alpha and Its Paralog CK2 alpha '. Pharmaceuticals, 10 (4). BASEL: MDPI. ISSN 1424-8247

الاتاحة: https://kups.ub.uni-koeln.de/20876/

المؤلفون: Jabor Gozzi, Gustavo, Bouaziz, Zouhair, Winter, Evelyn, Daflon-Yunes, Nathalia, Aichele, Dagmar, Nacereddine, Abdelhamib, Marminon, Christelle, Valdameri, Glaucio, Zeinyeh, Wael, Bollacke, Andre, Guillon, Jean, Lacoudre, Aline, Pinaud, Noël, Cadena, Silvia M, Jose, Joachim, Le Borgne, Marc, Di Pietro, Attilio

المساهمون: Bases moléculaires et structurales des systèmes infectieux (BMSSI), Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon-Centre National de la Recherche Scientifique (CNRS), Biomolécules Cancer et Chimiorésistances (B2C), Université de Lyon-Université de Lyon, Institut für Pharmazeutische und Medizinische Chemie, Westfälische Wilhelms-Universität Münster = University of Münster (WWU)

المصدر: ISSN: 0022-2623.

مصطلحات موضوعية: 2-b]indoles, indeno[1, protein kinase CK2, ABCG2, [CHIM.THER]Chemical Sciences/Medicinal Chemistry, [CHIM.CRIS]Chemical Sciences/Cristallography, [SDV.BBM]Life Sciences [q-bio]/Biochemistry, Molecular Biology, [SDV.BC]Life Sciences [q-bio]/Cellular Biology, [SDV.SP]Life Sciences [q-bio]/Pharmaceutical sciences

Relation: hal-01174925; https://hal.science/hal-01174925

الاتاحة: https://hal.science/hal-01174925
https://doi.org/10.1021/jm500943z