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1
المؤلفون: Chi-Yuan Chou, Chiao Che Chen, Yau-Hung Chen, David C. Moses, Chao Hsiung Lin, Hsu Feng Chu, Ying Chieh Tsai
المصدر: Antiviral Research
مصطلحات موضوعية: 0301 basic medicine, Alpha coronavirus, Protein Conformation, medicine.medical_treatment, viruses, CoV, coronavirus, Coronavirus Papain-Like Proteases, medicine.disease_cause, 6MP, 6-mercaptopurine, law.invention, PEDV, porcine epidemic diarrhea virus, chemistry.chemical_compound, SV, sedimentation velocity, USP, ubiquitin-specific protease, law, βME, β-mercaptoethanol, Papain, Noncompetitive inhibition, Coronavirus, Attenuated vaccine, PLpro, papain-like protease, biology, PEDV, 6-Thioguanine, Recombinant Proteins, Molecular Docking Simulation, Diarrhea, Recombinant DNA, PL2pro, papain-like protease 2, Ubl, ubiquitin-like, medicine.symptom, Coronavirus Infections, Proteases, DUB, deubiquitinating, Antiviral Agents, Article, 03 medical and health sciences, Virology, medicine, nsp, non-structural protein, SARS, severe acute respiratory syndrome, Thioguanine, Pharmacology, Protease, Binding Sites, Porcine epidemic diarrhea virus, MERS, Middle East respiratory syndrome, biology.organism_classification, PL1pro, papain-like protease 1, Ub-AFC, ubiquitin-7-amino-4-trifluoro-methyl-coumarin, Papain-like protease, Kinetics, 030104 developmental biology, chemistry, AUC, The abbreviations used are analytical ultracentrifugation, 6TG, 6-thioguanine
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2
المؤلفون: Dengke Tian, Liang Xin, Minge Wan, Xie Xiaolin, Zhang Dezhu, Wenqiang Cao, Liang Chengyuan, Liu Yuzhi, Li Han, Hong Liu, Xueqi Fu
المصدر: Biomedicine & Pharmacotherapy
Biomedicine & Pharmacotherapy, Vol 137, Iss, Pp 111313-(2021)مصطلحات موضوعية: 0301 basic medicine, Coronaviruses, medicine.medical_treatment, viruses, Review, Pharmacology, chemistry.chemical_compound, 0302 clinical medicine, nsps, Non-structural proteins, Chloroquine, Medicine, CoV, Coronavirus, CQ, Chloroquine, HA, Haemagglutinin, Molecular Targeted Therapy, Enzyme Inhibitors, DAAs, Direct-acting antiviral agents, biology, FDA, US Food and Drug Administration, Therapies, Investigational, HTAs, Host-targeting antivirals, MERS-CoV, Middle East respiratory syndrome coronavirus, General Medicine, Small molecule, PIP2, Phosphatidylinositol 4,5-bisphosphate, RMP, Ribavirin monophosphate, IFN, Interferon, N, Nucleocapsid protein, COVID-19, 2019 Coronavirus disease, HIV, Human immunodeficiency virus, RBV, Ribavirin, NIAID, National Institute of Allergy and Infectious Diseases, 030220 oncology & carcinogenesis, 6MP, 6-Mercaptopurine, BSAs, Broad-spectrum antiviral drugs, RDP, Ribavirin diphosphate, EBOV, Ebola virus, Transmembrane serine protease (TMPRSS2), GTP, Guanosine triphosphate, medicine.drug, 3CLpro, 3C-Like protease, DHODH, Dihydroorotate dehydrogenase, 6TG, 6-Thioguanine, Papain-like protease (PLpro), TGN, Trans-Golgi network, RM1-950, Favipiravir, TMPRSS2, HyCoSuL, Hybrid Combinatorial Substrate Library, Antiviral Agents, PP2A, Protein phosphatase 2A, SARS-CoV, Severe acute respiratory syndrome coronavirus, WHO, World Health Organization, CPE, Cytopathic effect, PLpro, Papain-like protease, 03 medical and health sciences, EUA, Emergency use authorization, IRF3, Interferon regulatory factor 3, SAR, Structure-activity relationship, ACE2, Angiotensin-converting enzyme 2, S, Spike protein, SKP2, S-Phase kinase-associated protein 2, Humans, RdRp, RNA-dependent RNA polymerase, RTP, Ribavirin triphosphate, BECN1, Beclin1, ComputingMethodologies_COMPUTERGRAPHICS, Serine protease, SARS-CoV-2, Severe acute respiratory syndrome coronavirus 2, Protease, HC, QHydroxychloroquine, business.industry, SARS-CoV-2, Ribavirin, fungi, COVID-19, PC, Pro-protein convertase, DHO, Dihydroorotate, M, Membrane protein, RNA-dependent RNA polymerase (RdRp), COVID-19 Drug Treatment, AMPK, AMP-activated protein kinase, CMK, Decanoyl-RVKR-chloromethylketone, Mpro, Main protease, 030104 developmental biology, chemistry, 3C-like protease (3CLpro), E, Envelope protein, biology.protein, Dihydroorotate dehydrogenase, GM1, Monosialotetrahexosylganglioside 1, LPV/r, Lopinavir/ritonavir, Therapeutics. Pharmacology, ELs, Endolysosomes, business, IMPDH, Inosine monophosphate dehydrogenase
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3
المؤلفون: Min-Han Lin, Chiao-Yin Sun, Shu-Chun Cheng, Wei Yi Chen, Kai-Wen Cheng, Chi-Yuan Chou, I-Hsin Cheng, Shang-Ju Chuang
المصدر: Antiviral Research
مصطلحات موضوعية: Models, Molecular, viruses, medicine.medical_treatment, CoV, coronavirus, 6MP, 6-mercaptopurine, medicine.disease_cause, Cysteine Proteases, Interferon, MERS-CoV papain-like protease, DUB, deubiquitination, Synergistic inhibition, Ub, ubiquitin, Coronavirus 3C Proteases, PLpro, papain-like protease, Thiopurine methyltransferase, biology, Mercaptopurine, 6-Thioguanine, virus diseases, Drug Synergism, respiratory system, Cysteine Endopeptidases, Immunosuppressive drug, Severe acute respiratory syndrome-related coronavirus, Middle East Respiratory Syndrome Coronavirus, Deubiquitination, medicine.drug, 6-Mercaptopurine, Middle East respiratory syndrome coronavirus, medicine.drug_class, Cysteine Proteinase Inhibitors, AFC, 7-amino-4-trifluoro-methylcoumarin, Antiviral Agents, Article, Mycophenolic acid, Viral Proteins, Virology, medicine, SARS, severe acute respiratory syndrome, Thioguanine, Pharmacology, Protease, MERS, Middle East respiratory syndrome, biochemical phenomena, metabolism, and nutrition, respiratory tract diseases, NEM, N-ethylmaleimide, biology.protein, Antiviral drug, 6TG, 6-thioguanine
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4
المؤلفون: Chi-Yuan Chou, Hsing Pang Hsieh, Yu-San Han, Chia Hui Chien, Boris Turk, Xin Chen, Mojca Trstenjak Prebanda, Gu-Gang Chang
المصدر: Biochemical Pharmacology
مصطلحات موضوعية: 6-Mercaptopurine, Proteases, Inhibitor, medicine.medical_treatment, CoV, coronavirus, DUB, deubiquitination enzyme, Biology, 6MP, 6-mercaptopurine, medicine.disease_cause, FRET, fluorescence resonance energy transfer, Biochemistry, Article, Viral Proteins, medicine, Protease Inhibitors, SARS, severe acute respiratory syndrome, AMC, 7-amino-4-methylcoumarin, Thioguanine, Coronavirus 3C Proteases, Coronavirus, Pharmacology, Cathepsin, chemistry.chemical_classification, Protease, Mercaptopurine, Severe acute respiratory syndrome coronavirus, 6-Thioguanine, Papain-like proteinase 2, Cysteine protease, Cysteine Endopeptidases, Enzyme, Severe acute respiratory syndrome-related coronavirus, chemistry, 3CLpro, 3-chymotrypsin-like protease, Docking (molecular), PLpro, papain-like proteinase 2, Pharmacophore, 6TG, 6-thioguanine
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5Academic Journal
المؤلفون: Deswal, Shivani, Srivastava, Anshu
المصدر: J Clin Exp Hepatol ; ISSN:0973-6883 ; Volume:7 ; Issue:1
مصطلحات موضوعية: 6-MTIMP, 6-methyl thioinosine monophosphate, 6MMP, 6-methyl mercaptopurine, 6MP, 6-mercaptopurine, 6TG, 6-thioguanine, AIH, autoimmune hepatitis, ANA, antinuclear antibody, AZA, azathioprine, HGPRT, hypoxanthine guanine phosphoribosyl transferase, IBD, inflammatory bowel disease, IgG, immunoglobulin G, LC, liver cytosol, LKM, liver kidney microsomal, PBC, primary biliary cirrhosis, PSC, primary sclerosing cholangitis, SMA, smooth muscle antibody, TIMP, thioinosine monophosphate, TPMT, thiopurine methyltransferase, XO, xanthine oxidase, allopurinol, autoimmune hepatitis, azathioprine, hepatotoxicity, overlap syndrome
Relation: https://doi.org/10.1016/j.jceh.2017.01.115; https://pubmed.ncbi.nlm.nih.gov/28348471; https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5357743/