المؤلفون: Lucia Sofrankova, Jana Spaldova, Pavol Stefik, Branislav Pavilek, Dusan Bortnak, Lucia Pavlikova, Ivana Zidekova, Daniel Vegh, Viktor Milata, Albert Breier, Zdena Sulova

المصدر: European Journal of Medicinal Chemistry Reports, Vol 13, Iss , Pp 100246- (2025)

مصطلحات موضوعية: 5-Aminopyrazoles, Cancer, Cell death, P-glycoprotein, Pharmacy and materia medica, RS1-441, Other systems of medicine, RZ201-999

Relation: http://www.sciencedirect.com/science/article/pii/S2772417425000020; https://doaj.org/toc/2772-4174; https://doaj.org/article/bf69d371f88e4bee9ed53481f3a376e9

الاتاحة: https://doi.org/10.1016/j.ejmcr.2025.100246
https://doaj.org/article/bf69d371f88e4bee9ed53481f3a376e9

المؤلفون: Federica Rapetti, Andrea Spallarossa, Eleonora Russo, Debora Caviglia, Carla Villa, Bruno Tasso, Maria Grazia Signorello, Camillo Rosano, Erika Iervasi, Marco Ponassi, Chiara Brullo

المصدر: Molecules, Vol 29, Iss 10, p 2298 (2024)

مصطلحات موضوعية: 5-aminopyrazoles, MTT test, anti-cancer activity, DPPH, ROS, druglike properties, Organic chemistry, QD241-441

Relation: https://www.mdpi.com/1420-3049/29/10/2298; https://doaj.org/toc/1420-3049; https://doaj.org/article/f972d7ba951b4953b48e4c2552e77869

الاتاحة: https://doi.org/10.3390/molecules29102298
https://doaj.org/article/f972d7ba951b4953b48e4c2552e77869

المؤلفون: Chiara Brullo, Debora Caviglia, Andrea Spallarossa, Silvana Alfei, Scott G. Franzblau, Bruno Tasso, Anna Maria Schito

المصدر: Pharmaceutics; Volume 14; Issue 9; Pages: 1770

مصطلحات موضوعية: pyrazole, 5-aminopyrazoles, antibacterial activity, Gram-positive species, Staphylococcus genus, in silico pharmacokinetic properties prediction

وصف الملف: application/pdf

Relation: Biopharmaceutics; https://dx.doi.org/10.3390/pharmaceutics14091770

الاتاحة: https://doi.org/10.3390/pharmaceutics14091770

المؤلفون: Abdallah AEM, Elgemeie GH

المصدر: Drug Design, Development and Therapy, Vol Volume 12, Pp 1785-1798 (2018)

مصطلحات موضوعية: Pyrazolo[1, 5-a]pyrimidines, 5-aminopyrazoles, 2-(hydroxymethylene)-1-cycloalkanones, 2-formylcycloalkanones, antimicrobial, docking studies., Therapeutics. Pharmacology, RM1-950

وصف الملف: electronic resource

Relation: https://www.dovepress.com/design-synthesis-docking-and-antimicrobial-evaluation-of-some-novel-py-peer-reviewed-article-DDDT; https://doaj.org/toc/1177-8881

URL الوصول: https://doaj.org/article/c30418a6d5e547f9b477d512bb2cb8fe

المؤلفون: Ranjana Aggarwal, Suresh Kumar

المصدر: Beilstein Journal of Organic Chemistry, Vol 14, Iss 1, Pp 203-242 (2018)

مصطلحات موضوعية: 5-aminopyrazoles, fused pyrazole derivatives, pyrazolopyridines, pyrazolopyrimidines, pyrazolotriazines, Science, Organic chemistry, QD241-441

وصف الملف: electronic resource

Relation: https://doaj.org/toc/1860-5397

URL الوصول: https://doaj.org/article/aa818b5e941f45b497e1a83897e96399

المؤلفون: Vladimir A. Kokorekin, Sergey V. Neverov, Vera N. Kuzina, Vladimir A. Petrosyan

المصدر: Molecules; Volume 25; Issue 18; Pages: 4169

مصطلحات موضوعية: thiocyanate group, 5-aminopyrazoles, 1,3-dicarbonyl compounds, pyrazolo[1,5- a ]pyrimidines, anodic C–H thiocyanation, condensation, cyclic voltammetry

جغرافية الموضوع: agris

وصف الملف: application/pdf

Relation: Organic Chemistry; https://dx.doi.org/10.3390/molecules25184169

الاتاحة: https://doi.org/10.3390/molecules25184169

المؤلفون: Mario A. Macías, Jessica Orrego-Hernández, Jaime Portilla

المصدر: Acta Crystallographica Section E: Crystallographic Communications, Vol 72, Iss 11, Pp 1672-1674 (2016)

مصطلحات موضوعية: crystal structure, pharmaceutical compound, 5-aminopyrazoles, nucleophilic substitution, hydrogen bonding, Crystallography, QD901-999

وصف الملف: electronic resource

Relation: http://scripts.iucr.org/cgi-bin/paper?S2056989016017187; https://doaj.org/toc/2056-9890

URL الوصول: https://doaj.org/article/28bb0c2b5ce342abb4376c18819f22df

المؤلفون: Zemlyana, N. I., Karnozhitska, T. M., Pavlovska, T. L., Mazepa, O. V., Musatov, V. I., Lipson, V. V.

المصدر: Журнал органічної та фармацевтичної хімії; Том 16 № 4(64) (2018); 3-10 ; Journal of Organic and Pharmaceutical Chemistry; Vol. 16 No. 4(64) (2018); 3-10 ; Журнал органической и фармацевтической химии; Том 16 № 4(64) (2018); 3-10 ; 2518-1548 ; 2308-8303

مصطلحات موضوعية: pyrazolo[3, 4-b]pyridine-4-spiroindolinones, 3-(5-aminopyrazol-4-yl)-3-hydroxy-2-oxindolines, isatins, 5-aminopyrazoles, 2-dimethyl-1, 3-dioxane-4, 6-dione, domino-reactions, UDC, 547.859.1, пиразоло[3, 4-b]пиридин-4-спироиндолиноны, 3-(5-аминопиразол-4-ил)-3-гидрокси-2-оксиндолины, изатины, 5-аминопиразолы, 2-диметил-1, 3-диоксан-4, 6-дион, домино-реакции, УДК, піразоло[3, 4-b]піридин-4-спіроіндолінони, 3-(5-амінопіразол-4-іл)-3-гідрокси-2-оксіндоліни, ізатини, 5-амінопіразоли, 3-діоксан-4, 6-діон, доміно-реакції

Time: 2

وصف الملف: application/pdf

Relation: http://ophcj.nuph.edu.ua/article/view/ophcj.18.950/150323; http://ophcj.nuph.edu.ua/article/view/ophcj.18.950

الاتاحة: http://ophcj.nuph.edu.ua/article/view/ophcj.18.950
https://doi.org/10.24959/ophcj.18.950

المؤلفون: Lozano Oviedo, John Jair

المساهمون: Cuervo Prado, Paola Andrea, Grupo de Estudios en Síntesis y Aplicaciones de Compuestos Heterocíclicos (Gesach)

المصدر: Repositorio UN
Universidad Nacional de Colombia
instacron:Universidad Nacional de Colombia

مصطلحات موضوعية: Electron-rich olefins, olefinas ricas en electrones, síntesis, Química orgánica-Síntesis, Multicomponent, Compuestos heterocíclicos, 5-aminopirazoles, Pyrazolopyridine, 5-aminopyrazoles, 540 - Química y ciencias afines, Microwave reaction, pirazolopiridinas, Heterocyclic Compounds, in silico, Organic compounds-Synthesis, GABA-A receptor, receptor GABA-A, microondas

وصف الملف: 143 páginas; application/pdf

URL الوصول: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::2dc7796ce2012b14f906b99f0886ab68
https://repositorio.unal.edu.co/

المؤلفون: Ranjana Aggarwal, Vinod Kumar, Rajiv Kumar, Shiv P. Singh

المصدر: Beilstein Journal of Organic Chemistry, Vol 7, Iss 1, Pp 179-197 (2011)

مصطلحات موضوعية: alkylidenemalononitriles, 5-aminopyrazoles, hydrazines, β-ketonitriles, malononitriles, Science, Organic chemistry, QD241-441

وصف الملف: electronic resource

Relation: https://doaj.org/toc/1860-5397

URL الوصول: https://doaj.org/article/28f1eef4c17f474c8050c92df8a133d2

المؤلفون: Lozano Oviedo, John Jair

المساهمون: Cuervo Prado, Paola Andrea, Grupo de Estudios en Síntesis y Aplicaciones de Compuestos Heterocíclicos (Gesach)

مصطلحات موضوعية: 540 - Química y ciencias afines, Compuestos heterocíclicos, Química orgánica-Síntesis, Heterocyclic Compounds, Organic compounds-Synthesis, in silico, pirazolopiridinas, microondas, receptor GABA-A, síntesis, 5-aminopirazoles, olefinas ricas en electrones, 5-aminopyrazoles, Pyrazolopyridine, Electron-rich olefins, Multicomponent, Microwave reaction, GABA-A receptor

وصف الملف: 143 páginas; application/pdf

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DOCK 6: Impact of New Features and Current Docking Performance. J. Comput. Chem. 2015, 36 (15), 1132–1156. https://doi.org/10.1002/JCC.23905.; LADIN, J. J. H.; Fabian Orozco López. DISEÑO, SÍNTESIS Y CARACTERIZACIÓN DE COMPUESTOS ESPIROTIAZAHETEROCÍCLICOS CON POTENCIAL ACTIVIDAD SOBRE SISTEMA NERVIOSO CENTRAL (SNC), Universidad Nacional de Colombia, 2019.; Bamoniri, A.; Mirjalili, B. B. F.; Jafari, A. A.; Abasaltian, F. Synthesis of 1,3,5-Tri-Substituted Pyrazoles Promoted by P2O5.SiO2. Iran. J. Catal. 2012, 2 (2), 75–78. https://doi.org/10.31857/s042485702109005x.; https://repositorio.unal.edu.co/handle/unal/82230; Universidad Nacional de Colombia; Repositorio Institucional Universidad Nacional de Colombia; https://repositorio.unal.edu.co/

الاتاحة: https://repositorio.unal.edu.co/handle/unal/82230
https://repositorio.unal.edu.co/

المؤلفون: Ashraf HASSAN, Taghrid HAFEZ, Souad OSMAN

المصدر: Scientia Pharmaceutica; Volume 83; Issue 1; Pages: 27-39

مصطلحات موضوعية: N -Substituted cyanoacetamide, Ketene N, S -acetals, Pyrazolo[1,5- a ]pyrimidines, 5-Aminopyrazoles, Cytotoxic activity

وصف الملف: application/pdf

Relation: https://dx.doi.org/10.3797/scipharm.1409-14

الاتاحة: https://doi.org/10.3797/scipharm.1409-14

المؤلفون: Vera N Kuzina, S. V. Neverov, Vladimir A. Petrosyan, Vladimir A. Kokorekin

المصدر: Molecules, Vol 25, Iss 4169, p 4169 (2020)
Molecules
Volume 25
Issue 18

مصطلحات موضوعية: Pyrimidine, Pharmaceutical Science, Ring (chemistry), 5-aminopyrazoles, Analytical Chemistry, lcsh:QD241-441, chemistry.chemical_compound, Thiocyanate ion, lcsh:Organic chemistry, Drug Discovery, Polymer chemistry, 1,3-dicarbonyl compounds, pyrazolo[1,5-a]pyrimidines, thiocyanate group, Physical and Theoretical Chemistry, Organic Chemistry, Condensation, Chemical condensation, Acceptor, cyclic voltammetry, condensation, chemistry, Chemistry (miscellaneous), Molecular Medicine, Cyclic voltammetry, anodic C–H thiocyanation

وصف الملف: application/pdf

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::19e26a8f9b4450863e48dbf0df414281
https://www.mdpi.com/1420-3049/25/18/4169

المؤلفون: Vladimir A, Kokorekin, Sergey V, Neverov, Vera N, Kuzina, Vladimir A, Petrosyan

المصدر: Molecules

مصطلحات موضوعية: Molecular Structure, Chemistry Techniques, Synthetic, Carbon, Electrolysis, Article, 5-aminopyrazoles, cyclic voltammetry, pyrazolo[1,5-a]pyrimidines, Structure-Activity Relationship, condensation, Pyrimidines, 1,3-dicarbonyl compounds, Electrochemistry, Pyrazoles, thiocyanate group, anodic C–H thiocyanation, Electrodes, Thiocyanates, Hydrogen

URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::df42979bb61d64ac522db6c7a79af764
https://pubmed.ncbi.nlm.nih.gov/32933044

المؤلفون: Hashmi, I.A., Feist, H., Michalik, M., Reinke, H., Peseke, K.

مصطلحات موضوعية: Reversed' C-Nucleoside Analogues, 5-Aminopyrazoles, Benzo[4,5]imidazo[1,2-a]pyridine, Pyrazolo[1,5-a]pyrimidines, Pyrimidines

Time: 540

وصف الملف: application/pdf; text/plain; charset=utf-8

الاتاحة: https://doi.org/10.34657/4171
https://oa.tib.eu/renate/handle/123456789/5542

المؤلفون: Suresh Kumar, Ranjana Aggarwal

المصدر: Beilstein Journal of Organic Chemistry
Beilstein Journal of Organic Chemistry, Vol 14, Iss 1, Pp 203-242 (2018)

مصطلحات موضوعية: 010405 organic chemistry, Chemistry, Condensation, Organic Chemistry, Review, fused pyrazole derivatives, 010402 general chemistry, 01 natural sciences, Combinatorial chemistry, 5-aminopyrazoles, 0104 chemical sciences, lcsh:QD241-441, lcsh:Organic chemistry, Organic reaction, pyrazolopyrimidines, lcsh:Q, lcsh:Science, pyrazolopyridines, pyrazolotriazines

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8e06fe785cdc439f75ce1f51bb93c24a
http://europepmc.org/articles/PMC5789427

المؤلفون: Amira E M, Abdallah, Galal H, Elgemeie

المصدر: Drug Design, Development and Therapy

مصطلحات موضوعية: Antifungal Agents, Molecular Structure, 2-(hydroxymethylene)-1-cycloalkanones, Proton Magnetic Resonance Spectroscopy, Cycloparaffins, docking studies, Gram-Positive Bacteria, 2-formylcycloalkanones, Mass Spectrometry, 5-aminopyrazoles, Anti-Bacterial Agents, pyrazolo[1,5-a]pyrimidines, Molecular Docking Simulation, Structure-Activity Relationship, antibacterial, Pyrimidines, Disk Diffusion Antimicrobial Tests, Drug Design, Candida albicans, Gram-Negative Bacteria, Spectroscopy, Fourier Transform Infrared, Pyrazoles, antifungal, Aspergillus flavus, Original Research

URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::940e2d8555c26ba098bda81b914f8406
https://pubmed.ncbi.nlm.nih.gov/29950813

المؤلفون: Jessica Orrego-Hernández, Jaime Portilla, Mario A. Macías

المصدر: Acta Crystallographica Section E: Crystallographic Communications, Vol 72, Iss 11, Pp 1672-1674 (2016)
Acta Crystallographica Section E: Crystallographic Communications

مصطلحات موضوعية: crystal structure, Crystal structure, Dihedral angle, Pyrazole, 010402 general chemistry, 01 natural sciences, Microwave assisted, pharmaceutical compound, 5-aminopyrazoles, Caesium carbonate, Research Communications, Catalysis, lcsh:Chemistry, chemistry.chemical_compound, Polymer chemistry, Nucleophilic substitution, Organic chemistry, General Materials Science, Quantitative Biology::Biomolecules, 010405 organic chemistry, Chemistry, Hydrogen bond, General Chemistry, hydrogen bonding, Condensed Matter Physics, 0104 chemical sciences, lcsh:QD1-999, 5-amino­pyrazoles, nucleophilic substitution

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::59b5c2a312dd5b995a817ce486939a46
https://doi.org/10.1107/s2056989016017187

المؤلفون: 劉柏麟, Po-Lin Liu

المساهمون: 藥物化學研究所碩士班

مصطلحات موضوعية: Vilsmeier反應, 5-氨基?紹, ?紹?[3,4-d]嘧啶, 甲?謋??承I, Vilsmeier reaction, 5-Aminopyrazoles, Pyrazolo[3,4-d]pyrimidine, Formamidine, Formamide

Relation: http://ir.cmu.edu.tw/ir/handle/310903500/54329; http://ir.cmu.edu.tw/ir/bitstream/310903500/54329/2/index.html; http://ir.cmu.edu.tw/ir/bitstream/310903500/54329/3/index.html; http://ir.cmu.edu.tw/ir/bitstream/310903500/54329/1/index.html

الاتاحة: http://ir.cmu.edu.tw/ir/handle/310903500/54329
http://ir.cmu.edu.tw/ir/bitstream/310903500/54329/2/index.html
http://ir.cmu.edu.tw/ir/bitstream/310903500/54329/3/index.html
http://ir.cmu.edu.tw/ir/bitstream/310903500/54329/1/index.html

المؤلفون: Chang, Chun-Hsi, 蔡建鈞, Tsai, Henry Jan-Jen, Huang, Yu-Ying, Lin, Hui-Yi, Wang, Li-Ya, Wu, Tian-Shung, Wong, Fung Fuh

المساهمون: 保健營養生技學系

مصطلحات موضوعية: Vilsmeier reaction, 5-Aminopyrazoles, Pyrazolo[3,4-d]pyrimidine, Formamidine, Formamide

Relation: TETRAHEDRON, 69(4):1378-1386.; http://asiair.asia.edu.tw/ir/handle/310904400/25284; http://asiair.asia.edu.tw/ir/bitstream/310904400/25284/1/index.html

الاتاحة: http://asiair.asia.edu.tw/ir/handle/310904400/25284
http://asiair.asia.edu.tw/ir/bitstream/310904400/25284/1/index.html