نتائج البحث - "10727388 - Petzer, Jacobus Petrus"

1

Electronic Resource

The evaluation of 1-tetralone and 4-chromanone derivatives as inhibitors of monoamine oxidase

المؤلفون: 12264954 - Petzer, Anél, 10727388 - Petzer, Jacobus Petrus, 12902608 - Legoabe, Lesetja Jan, 21695814 - N'Da, Clarina Ilara, 23496959 - Cloete, Stephanus J., Cloete, Stephanus J., N'Da, Clarina I., Legoabe, Lesetja J., Petzer, Anél, Petzer, Jacobus P.

مصطلحات الفهرس: 1-Tetralone, 4-Chromanone, Monoamine oxidase, Inhibition, Parkinson’s disease, Article

URL: http://hdl.handle.net/10394/35833

View record in OAIster

2

Electronic Resource

Synthesis and evaluation of 7-azaindole derivatives bearing benzocycloalkanone motifs as protein kinase inhibitors

المؤلفون: 10727388 - Petzer, Jacobus Petrus, 12902608 - Legoabe, Lesetja Jan, 25159194 - Beteck, Richard Mbi, 27836576 - Qhobosheane, Malikotsi A., Qhobosheane, Malikotsi A., Legoabe, Lesetja J., Petzer, Jacobus P., Beteck, Richard M., Josselin, Béatrice

مصطلحات الفهرس: 7-Azaindole, Benzocycloalkanone, Protein kinase, Structure-activity relationship, Haspin, CDK9/CyclinT, Dual inhibitor, Oncology, Article

URL: http://hdl.handle.net/10394/34563
https://www.sciencedirect.com/science/article/pii/S0968089620302820
https://doi.org/10.1016/j.bmc.2020.115468

View record in OAIster

3

Electronic Resource

Design, synthesis and evaluation of 3-hydroxypyridin-4-ones as inhibitors of catechol-O-methyltransferase

المؤلفون: 10727388 - Petzer, Jacobus Petrus, 12264954 - Petzer, Anél, 10948724 - Lourens, Anna Catharina U., 22155600 - De Beer, Johannie, De Beer, Johannie, Petzer, Jacobus P., Lourens, Anna C.U., Petzer, Anél

مصطلحات الفهرس: 3-Hydroxypyridin-4-one, Catechol-O-methyltransferase, COMT, Inhibition, Parkinson’s disease, Article

URL: http://hdl.handle.net/10394/34450
https://link.springer.com/article/10.1007/s11030-020-10053-x
https://doi.org/10.1007/s11030-020-10053-x

View record in OAIster

4

Electronic Resource

The monoamine oxidase inhibition properties of C6-and N1-substituted 3-methyl-3,4-dihydroquinazolin-2(1H)-one derivatives

المؤلفون: 12264954 - Petzer, Anél, 10727388 - Petzer, Jacobus Petrus, 12902608 - Legoabe, Lesetja Jan, 22161333 - Marais, Lereze, Marais, Lereze, Petzer, Anél, Pelzer, Jacobus P., Legoabe, Lesetja J.

مصطلحات الفهرس: Monoamine oxidase, MAO, Inhibition, Reversible, Quinazolinone, Article

URL: http://hdl.handle.net/10394/34845
https://link.springer.com/article/10.1007/s11030-019-09960-5
https://doi.org/10.1007/s11030-019-09960-5

View record in OAIster

5

Electronic Resource

Methylene blue analogues: in vitro antimicrobial minimum inhibitory concentrations and in silico pharmacophore modelling

المؤلفون: 10727388 - Petzer, Jacobus Petrus, 12264954 - Petzer, Anél, 10926542 - Bezuidenhout, Johannes Jacobus, 13061372 - Cloete, Theunis Theodorus, 24942847 - Thesnaar, Louis C., Thesnaar, Louis, Bezuidenhout, Jaco J., Petzer, Anél, Petzer, Jacobus P., Cloete, Theunis T.

مصطلحات الفهرس: Discovery Studio, Methylene blue, Antimicrobial activity, Common feature pharmacophore modelling, Article

URL: http://hdl.handle.net/10394/36475
https://www.sciencedirect.com/science/article/pii/S0928098720303912
https://doi.org/10.1016/j.ejps.2020.105603

View record in OAIster

6

Electronic Resource

The monoamine oxidase inhibition properties of C6- and N1-substituted 3-methyl-3,4-dihydroquinazolin-2(1H)-one derivatives

المؤلفون: 10727388 - Petzer, Jacobus Petrus, 12264954 - Petzer, Anél, 12902608 - Legoabe, Lesetja Jan, 22161333 - Marais, Lereze, Marais, Lereze, Petzer, Anél, Petzer, Jacobus P., Legoabe, Lesetja J.

مصطلحات الفهرس: Monoamine oxidase, MAO, Inhibition, Reversible, Quinazolinone, Neurodegenerative disorders, Article

URL: http://hdl.handle.net/10394/32503
https://link.springer.com/article/10.1007/s11030-019-09960-5
https://doi.org/10.1007/s11030-019-09960-5

View record in OAIster

7

Electronic Resource

The monoamine oxidase inhibition properties of C6-mono- and N3/C6-disubstituted derivatives of 4(3H)-quinazolinone

المؤلفون: 12902608 - Legoabe, Lesetja Jan, 12264954 - Petzer, Anél, 10727388 - Petzer, Jacobus Petrus, 27836576 - Qhobosheane, Malikotsi A., Qhobosheane, Malikotsi A., Legoabe, Lesetja J., Petzer, Anél, Petzer, Jacobus P.

مصطلحات الفهرس: Monoamine oxidase, MAO, Quinazolinone, Parkinson’s disease, Inhibition, Article

URL: http://hdl.handle.net/10394/31749

View record in OAIster

8

Electronic Resource

SAR and molecular mechanism studies of monoamine oxidase inhibition by selected chalcone analogs

المؤلفون: 10727388 - Petzer, Jacobus Petrus, 12264954 - Petzer, Anél, Shalaby, Raed, Petzer, Jacobus P., Petzer, Anél, Ashraf, Usman M., Atari, Ealla

مصطلحات الفهرس: Monoamine oxidase, Chalcone, Reversibility, Dopamine, mRNA, Article

URL: http://hdl.handle.net/10394/32266

View record in OAIster

9

Electronic Resource

Monoamine oxidase inhibition by selected dye compounds

المؤلفون: 10727388 - Petzer, Jacobus Petrus, 12264954 - Petzer, Anél, De Beer, Franciska, Petzer, Jacobus P., Petzer, Anél

مصطلحات الفهرس: Acridine orange, Darrow red, Inhibition, Methylene blue, Monoamine oxidase, Oxazine 170, Article

URL: http://hdl.handle.net/10394/34184

View record in OAIster

10

Electronic Resource

Novel monoamine oxidase inhibitors based on the privileged 2-imidazoline molecular framework

المؤلفون: 10727388 - Petzer, Jacobus Petrus, 12264954 - Petzer, Anél, 21639159 - Engelbrecht, Idalet, Shetnev, Anton, Petzer, Anél, Engelbrecht, Idalet, Petzer, Jacobus P., Osipyan, Angelina

مصطلحات الفهرس: Monoamine oxidase, MAO, Inhibition, Selective, 2-Imidazoline, Article

URL: http://hdl.handle.net/10394/31752
https://www.sciencedirect.com/science/article/pii/S0960894X18308837
https://doi.org/10.1016/j.bmcl.2018.11.018

View record in OAIster

11

Electronic Resource

4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis

المؤلفون: 10727388 - Petzer, Jacobus Petrus, 12264954 - Petzer, Anél, Secci, Daniela, Petzer, Anél, Petzer, Jacobus P., Carradori, Simone, Guglielmi, Paulo

مصطلحات الفهرس: (Thiazol-2-yl)hydrazone derivatives, Alzheimer’s disease, Parkinson’s disease, Selective, Monoamine oxidase, Inhibitor, Antioxidants, Molecular modelling, Article

URL: http://hdl.handle.net/10394/31905
https://doi.org/10.1080/14756366.2019.1571272

View record in OAIster

12

Electronic Resource

Development and validation of a HPLC electrochemical detection method to measure COMT activity as a tool in drug development

المؤلفون: 11775416 - Viljoen, Francois Petrus, 10060510 - Du Preez, Jan Lourens, 12264954 - Petzer, Anél, 10727388 - Petzer, Jacobus Petrus, 10204040 - Wessels, Johanna Christina, Viljoen, F.P., Du Preez, J.L., Petzer, A., Wessels, J.C., Petzer, J.

مصطلحات الفهرس: Article

URL: http://hdl.handle.net/10394/32498
https://www.ingentaconnect.com/contentone/govi/pharmaz/2019/00000074/00000005/art00003
https://doi.org/10.1691/ph.2019.8218

View record in OAIster

13

Electronic Resource

Synthesis and evaluation of 2-substituted 4(3H)-quinazolinone thioether derivatives as monoamine oxidase inhibitors

المؤلفون: 12264954 - Petzer, Anél, 10727388 - Petzer, Jacobus Petrus, 12902608 - Legoabe, Lesetja Jan, 27836576 - Qhobosheane, Malikotsi A., Qhobosheane, Malikotsi A., Petzer, Anél, Petzer, Jacobus P., Legoabe, Lesetja J.

مصطلحات الفهرس: Monoamine oxidase, MAO, Inhibition, Reversible, Quinazolinone, Parkinson’s disease, Article

URL: http://hdl.handle.net/10394/31518

View record in OAIster

14

Electronic Resource

Methylene blue analogues with marginal monoamine oxidase inhibition retain antidepressant-like activity

المؤلفون: 21219079 - Delport, Anzelle, 11083417 - Harvey, Brian Herbert, 12264954 - Petzer, Anél, 10727388 - Petzer, Jacobus Petrus, Delport, Anzelle, Harvey, Brian H., Petzer, Anél, Petzer, Jacobus P.

مصطلحات الفهرس: Azure B, Depression, Forced swim test, Inhibition, Mitochondrial electron transport, Nitric oxide, Article

URL: http://hdl.handle.net/10394/31677

View record in OAIster

15

Electronic Resource

Nitrocatechol derivatives of chalcone as inhibitors of monoamine oxidase and Catechol-O-Methyltransferase

المؤلفون: 21639159 - Engelbrecht, Idalet, 10727388 - Petzer, Jacobus Petrus, 12264954 - Petzer, Anél, Engelbrecht, Idalet, Petzer, Jacobus P., Petzer, Anél

مصطلحات الفهرس: Catechol-O-methyltransferase, Chalcone, COMT, Inhibition, MAO, Monoamine oxidase, Multi-target-directed, Parkinson's disease, Article

URL: http://hdl.handle.net/10394/30746
http://www.eurekaselect.com/161603

View record in OAIster

16

Electronic Resource

Synthesis and in vitro evaluation of 2-heteroarylidene-1-tetralone derivatives as monoamine oxidase inhibitors

المؤلفون: 12902608 - Legoabe, Lesetja Jan, 10727388 - Petzer, Jacobus Petrus, 12264954 - Petzer, Anél, Amakali, Klaudia T., Legoabe, Lesetja J., Petzer, Anél, Petzer, Jacobus P.

مصطلحات الفهرس: Monoamine oxidase, Inhibition, Parkinson’s disease, Alzheimer’s disease, Heteroarylidene-1-tetralone, 2-Benzylidene-1-tetralone, Article

URL: http://hdl.handle.net/10394/31725

View record in OAIster

17

Electronic Resource

An investigation of the monoamine oxidase inhibition properties of pyrrolo[3,4‐f]indole‐5,7‐dione and indole‐5,6‐dicarbonitrile derivatives

المؤلفون: 12264954 - Petzer, Anél, 10727388 - Petzer, Jacobus Petrus, 21639159 - Engelbrecht, Idalet, Chirkova, Zhanna, V., Petzer, Anél, Engelbrecht, Idalet, Petzer, Jacobus P., Kabanova, Mariya V.

مصطلحات الفهرس: Inhibition, Indole‐5,6‐dicarbonitriles, MAO, Monoamine oxidase, Pyrrolo[3,4‐ f]indole‐5,7‐diones, Article

URL: http://hdl.handle.net/10394/26879
https://onlinelibrary.wiley.com/doi/abs/10.1002/ddr.21425
https://doi.org/10.1002/ddr.21425

View record in OAIster

18

Electronic Resource

MAO inhibitors and their wider applications: a patent review

المؤلفون: 10727388 - Petzer, Jacobus Petrus, Carradori, Simone, Petzer, Jacques P., Secci, Daniela

مصطلحات الفهرس: Alzheimer’s disease, Depression, Multi-target inhibitors, Monoamine oxidase, Natural products, Parkinson’s disease, Article

URL: http://hdl.handle.net/10394/26560
https://www.tandfonline.com/doi/full/10.1080/13543776.2018.1427735
https://doi.org/10.1080/13543776.2018.1427735

View record in OAIster

19

Electronic Resource

Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents

المؤلفون: 12264954 - Petzer, Anél, 10727388 - Petzer, Jacobus Petrus, Carradori, Simone, Petzer, Anél, Petzer, Jacobus P., Ortuso, Francesco, Bagetta, Donatella

مصطلحات الفهرس: Dual-target-directed, Rational design, Thiazol-2-ylhydrazones, Parkinson's disease, Selective monoamine oxidase inhibitors, Selective cholinesterase inhibitors, Antioxidant agents, Article

URL: http://hdl.handle.net/10394/26436
https://www.sciencedirect.com/science/article/pii/S0223523417308528
https://doi.org/10.1016/j.ejmech.2017.10.050

View record in OAIster

20

Electronic Resource

Methylene blue and its analogues as antidepressant compounds

المؤلفون: 12264954 - Petzer, Anél, 10727388 - Petzer, Jacobus Petrus, 11083417 - Harvey, Brian Herbert, 21219079 - Delport, Anzelle, Delport, Anzelle, Harvey, Brian Herbert, Petzer, Anél, Petzer, Jacobus P.

مصطلحات الفهرس: Methylene blue, Depression, Monoamine oxidase, Nitric oxide synthase, mitochondrial function, Reactive oxygen species, Article

URL: http://hdl.handle.net/10394/25492
https://link.springer.com/article/10.1007/s11011-017-0081-6
https://doi.org/10.1007/s11011-017-0081-6

View record in OAIster

تنقيح النتائج