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1Academic Journal
المؤلفون: Singh, R., Bhardwaj, V. K., Das, P., Bhattacherjee, D., Zyryanov, G. V., Purohit, R.
المصدر: Computers in Biology and Medicine
مصطلحات موضوعية: 1,2,3-TRIAZOLE, FREE ENERGY LANDSCAPE, MD SIMULATION, MM-PBSA, UMBRELLA SAMPLING SIMULATION, BINDING ENERGY, DISEASES, FREE ENERGY, MOLECULAR DYNAMICS, DEVELOPMENT PROCESS, DRUG DEVELOPMENT, SAMPLING SIMULATION, STEERED MOLECULAR DYNAMICS SIMULATIONS, UMBRELLA SAMPLING, SARS, 1,2,3 TRIAZOLE DERIVATIVE, CORONAVIRUS 3C PROTEASE, CORONAVIRUS PROTEINASE INHIBITOR, 3C-LIKE PROTEINASE, SARS-COV-2, CYSTEINE PROTEINASE, PROTEINASE INHIBITOR, TRIAZOLE DERIVATIVE, VIRAL PROTEIN, ARTICLE, BINDING AFFINITY, CONTROLLED STUDY, DRUG DESIGN, DRUG PROTEIN BINDING, DRUG STABILITY
وصف الملف: application/pdf
Relation: Benchmarking the ability of novel compounds to inhibit SARS-CoV-2 main protease using steered molecular dynamics simulations / R. Singh, V. K. Bhardwaj, P. Das et al. // Computers in Biology and Medicine. — 2022. — Vol. 146. — 105572.; https://www.scopus.com/inward/record.uri?eid=2-s2.0-85129703595&doi=10.1016%2fj.compbiomed.2022.105572&partnerID=40&md5=a71ef4adcea6891ae533c65d414145e3; http://elar.urfu.ru/handle/10995/118366; 85129703595; 000804709400004
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2Academic Journal
المؤلفون: Filimonov, V. O., Dianova, L. N., Beryozkina, T. V., Mazur, D., Beliaev, N. A., Volkova, N. N., Ilkin, V. G., Dehaen, W., Lebedev, A. T., Bakulev, V. A.
المصدر: J. Org. Chem. ; Journal of Organic Chemistry
مصطلحات موضوعية: AROMATIC COMPOUNDS, CHLORINE COMPOUNDS, SODIUM AZIDE, 1 ,2 ,3-TRIAZOLES, AROMATIC AZIDES, ATOM ECONOMIC, ECO-FRIENDLY, ONE-POT REACTION, ROLE OF WATER, SULFONYL AZIDES, SULFONYL CHLORIDES, ENVIRONMENTAL PROTECTION, 1,2,3 TRIAZOLE DERIVATIVE, ALKALI, AZIDE, CHLORIDE, THIADIAZOLE DERIVATIVE, THIOACETAMIDE DERIVATIVE, WATER, ARTICLE, CATALYST, CHEMICAL REACTION, ONE POT SYNTHESIS, SYNTHESIS
وصف الملف: application/pdf
Relation: info:eu-repo/grantAgreement/RSF//18-13-00161; Water/Alkali-Catalyzed Reactions of Azides with 2-Cyanothioacetamides. Eco-Friendly Synthesis of Monocyclic and Bicyclic 1,2,3-Thiadiazole-4-carbimidamides and 5-Amino-1,2,3-triazole-4-carbothioamides / V. O. Filimonov, L. N. Dianova, T. V. Beryozkina et al. // Journal of Organic Chemistry. — 2019. — Vol. 84. — Iss. 21. — P. 13430-13446.; All Open Access, Green; http://elar.urfu.ru/handle/10995/111996; 85073120953
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3Academic Journal
المؤلفون: Kyriakis E., Karra A.G., Papaioannou O., Solovou T., Skamnaki V.T., Liggri P.G.V., Zographos S.E., Szennyes E., Bokor É., Kun S., Psarra A.-M.G., Somsák L., Leonidas D.D.
المصدر: Bioorganic and Medicinal Chemistry ; https://www.scopus.com/inward/record.uri?eid=2-s2.0-85076026403&doi=10.1016%2fj.bmc.2019.115196&partnerID=40&md5=35b2a3588f3b971c8cb05e27585c4267
مصطلحات موضوعية: 1,2,3 triazole derivative, c beta dextro glucopyranosyl thiazole derivative, glycogen phosphorylase, hydrogen, hyperglycemic agent, imidazole derivative, n beta dextro glucopyranosyl tetrazole, thiazole derivative, unclassified drug, enzyme inhibitor, sulfur, tetrazole derivative, Article, controlled study, drug design, drug potency, drug structure, drug synthesis, drug targeting, enzyme activity, enzyme inhibition, enzyme inhibitor complex, ex vivo study, Hep-G2 cell line, human, human cell, hydrogen bond, in vitro study, X ray crystallography, chemical structure
Relation: http://hdl.handle.net/11615/75572
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4
المؤلفون: Gilles Hanquet, Gabriela Addová, Juraj Dobiaš, Margaréta Vojtičková, Andrej Boháč, Rengul Cetin-Atalay, Deniz Yildirim
المصدر: European Journal of Medicinal Chemistry
مصطلحات موضوعية: Oxazole/1,2,3-triazole isosteric replacement, Molecular model, protein tyrosine kinase inhibitor, Protein Data Bank (RCSB PDB), 4 [4 [5 (ethylsulfonyl) 2 methoxyphenylamino] 1h 1,2,3 triazol 1 yl] 2 (pyridin 2 yl)phenol, VEGFR2 tyrosine kinase inhibition, CuACC Click chemistry, chemistry.chemical_compound, Drug Discovery, vasculotropin receptor 2, phosphatidylinositol 3 kinase, Oxazole, carcinoma cell line, Molecular Structure, Chemistry, 1,2,3 triazole derivative, General Medicine, unclassified drug, enzyme activity, PI3K/Akt pathway, Alkynes, click chemistry, Click chemistry, Cytotoxic activity in Huh-7 and Mahlavu, cytotoxicity, chemical reaction, liver cell carcinoma, Stereochemistry, Triazole, Antineoplastic Agents, Article, Structure-Activity Relationship, Cell Line, Tumor, Humans, Structure–activity relationship, controlled study, human, Ynamide, Binding site, Protein Kinase Inhibitors, Cell Proliferation, Pharmacology, Dose-Response Relationship, Drug, binding site, human cell, oxazole, Organic Chemistry, molecular docking, Triazoles, Amides, Vascular Endothelial Growth Factor Receptor-2, drug structure, concentration response, Docking (molecular), protein kinase B, drug synthesis, Click Chemistry, molecular model, Drug Screening Assays, Antitumor, hepatocellular carcinoma cell lines
وصف الملف: application/pdf
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5Academic Journal
المؤلفون: PIPPIONE, Agnese Chiara, DOSIO, Franco, DUCIME, ALEX, FEDERICO, ANTONELLA, MARTINA, Katia, SAINAS, STEFANO, BOSCHI, Donatella, LOLLI, Marco Lucio, Frølund, Bente, Gooyit, Major, Janda, Kim D.
المساهمون: Pippione, Agnese C, Dosio, Franco, Ducime, Alex, Federico, Antonella, Martina, Katia, Sainas, Stefano, Frølund, Bente, Gooyit, Major, Janda, Kim D., Boschi, Donatella, Lolli, Marco L.
مصطلحات موضوعية: Biochemistry, 1,2,3 triazole derivative, 4 hydroxy 1,2,3 triazole derivative, chitinase, enzyme inhibitor
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:000357786200009; volume:6; issue:7; firstpage:1285; lastpage:1292; numberofpages:8; journal:MEDCHEMCOMM; http://hdl.handle.net/2318/1544314; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-84936875091; http://www.rsc.org/Publishing/Journals/MD/About.asp
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6Academic Journal
المؤلفون: Bokor E., Kyriakis E., Solovou T.G.A., Koppány C., Kantsadi A.L., Szabó K.E., Szakács A., Stravodimos G.A., Docsa T., Skamnaki V.T., Zographos S.E., Gergely P., Leonidas D.D., Somsák L.
المصدر: Journal of Medicinal Chemistry ; https://www.scopus.com/inward/record.uri?eid=2-s2.0-85034949385&doi=10.1021%2facs.jmedchem.7b01056&partnerID=40&md5=a379c9e0ee780b4db4fcc07884628954
مصطلحات موضوعية: 1 (2' amino 2' deoxy beta dextro glucopyranosyl) 4 (2 naphthyl) 1,2,3 triazole, 1 (2' amino 2' deoxy beta dextro glucopyranosyl) 4 phenyl 1,2,3 triazole, 1,2,3 triazole derivative, 1,2,4 triazole derivative, 2 (2' amino 2' deoxy beta dexro glucopyranosyl) 4(5) (2 naphthyl)imidazole, 2 (2' amino 2' deoxy beta dextro glucopyranosyl) 4(5)phenyl imidazole, 2 (2' amino 2' deoxy beta dextro glucopyranosyl)benzimidazole, 2 (2' deoxy 2' phthalimido 3',4',6' tri o acetyl beta detro glucopyranosyl) 4(5) phenyl imidazole, 2 (2' deoxy 2' phthalimido 3',4',6' tri o acetyl beta dextro glucopyranosyl) 4(5) (2 naphthyl)imidazole, 2 (2' deoxy 2' phthalimido 3',4',6' tri o acetyl beta dextro glucopyranosyl)benzimidazole, 3 (2' amino 2' deoxy beta dextro glucopyranosyl) 5 (2 naphthyl) 1,2,4 triazole, 3 (2' amino 2' deoxy beta dextro glucopyranosyl) 5 phenyl 1,2,4 triazole, ethyl c (2 deoxy 2 phthalimido 3,4,6 tri o acetyl beta dextro glucopyranosyl)formimidate, glucosamine derivative, glycogen phosphorylase, glycosyltransferase inhibitor, heterocyclic compound, imidazole derivative, n (2 deoxy 2 phthalimido 3,4,6 tri o acetyl beta dextro glucopyranosylcarbonyl)benzenethiocarboxamide, n (2 deoxy 2 phthalimido 3,4,6 tri o acetyl beta dextro glucopyranosylcarbonyl)naphthalene 2 thiocarboxamide, unclassified drug, 2-(2'-amino-2'-deoxyglucopyranosyl)-4(5)-(2-naphthyl)imidazole, glucosamine, triazole derivative, allosteric site, animal tissue, Article, comparative study, competitive inhibition, controlled study
Relation: http://hdl.handle.net/11615/71804
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7
المؤلفون: Rishi Kumar, Nam Huan Khieu, Milan Bhasin, Harold C. Jarrell, Wei Zou, Michel Gilbert, Margaret Hsieh, Harold J. Jennings, Ravindranath Nasi
المصدر: Carbohydrate Research. 378:45-55
مصطلحات موضوعية: sialyltransferase, Hydrophobicity, Biochemistry, Nitrogen compounds, Analytical Chemistry, chemistry.chemical_compound, Biomimetic Materials, benzoic acid derivative, Sialyltransferease inhibitors>, Amide, binding affinity, Moiety, Enzyme Inhibitors, Sulfur compounds, enzyme inhibition, chemistry.chemical_classification, biology, Click chemistry, Chemistry, 1,2,3 triazole derivative, Cytidine, General Medicine, Amino acid, competitive inhibition, Synthesis (chemical), Amino acids, Hydrophobic and Hydrophilic Interactions, cytidine phosphate n acetylneuraminic acid, glycosylation, Stereochemistry, Sialyltransferase, Carboxylic acid, 1,2,3-Triazole, Sialic acids, Binding energy, Campylobacter jejuni, Hydrophobic effect, sulfanilamide, sulfonamide, Binding selectivity, phosphate, hydrogen bond, Bacteria, Carboxylic acids, Organic Chemistry, molecular docking, 2-Deoxy-2, Molecules, Sialyltransferases, cytidine, 2-Deoxy-2,3-dehydro-acetylneuraminic acid, Drug Design, molecular interaction, chemical structure, biology.protein
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8
المؤلفون: Stefano Sainas, Marco Lucio Lolli, Alex Ducime, Franco Dosio, Bente Frølund, Katia Martina, Major Gooyit, Kim D. Janda, Antonella Federico, Agnese Chiara Pippione, Donatella Boschi
مصطلحات موضوعية: Drug, Scaffold, Stereochemistry, media_common.quotation_subject, Carboxylic acid, Triazole, enzyme inhibitor, Pharmaceutical Science, Scaffold hopping, Ring (chemistry), Biochemistry, 4 hydroxy 1, chemistry.chemical_compound, Drug Discovery, Moiety, media_common, Pharmacology, chemistry.chemical_classification, Chemistry, Organic Chemistry, Combinatorial chemistry, Biochemistry, 1,2,3 triazole derivative, 4 hydroxy 1,2,3 triazole derivative, chitinase, enzyme inhibitor, chitinase, Molecular Medicine, 3 triazole derivative
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9
المصدر: Tetrahedron Letters. 50:5834-5837
مصطلحات موضوعية: biphenyl derivative, synthesis, Suzuki reaction, Stereochemistry, chemistry.chemical_element, carbenoid, Biochemistry, Medicinal chemistry, Catalysis, Ion, chemistry.chemical_compound, Bromide, Drug Discovery, bromine derivative, naphthalene derivative, catalysis, 1,2,3 triazole derivative, Aryl, Organic Chemistry, palladium complex, Pincer movement, reaction analysis, boronic acid derivative, chemistry, Carbene, Palladium
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10
المؤلفون: Duraikkannu Loganathan, Katuri J.V. Paul
المصدر: Tetrahedron Letters. 49:6356-6359
مصطلحات موضوعية: chemistry.chemical_classification, Chemistry, Organic Chemistry, Biochemistry, Cycloaddition, Catalysis, Glycolipid, Acetylation, Drug Discovery, Propargyl, 1,2,3 triazole derivative, amide, azide, cuprous ion, ether lipid, glucose, glycolipid, glycopyranosyl azide, n (beta glycopyranosyl)azidoacetamide, unclassified drug, acetylation, catalysis, cycloaddition, drug structure, lipogenesis, Click chemistry, Organic chemistry, Long chain, Alkyl
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11
المؤلفون: Shanmugam Rajasekar, Pazhamalai Anbarasan
المصدر: The Journal of organic chemistry. 79(17)
مصطلحات موضوعية: Antitumor activity, Molecular Structure, Organic Chemistry, chemistry.chemical_element, Antineoplastic Agents, Vinyl ether, Triazoles, Catalysis, 1 ,2 ,3-triazoles, Anti-tumor agents, Formal synthesis, Rhodium-catalyzed, Transannulation, Vinyl ethers, Rhodium, 1,2,3 triazole derivative, antineoplastic agent, neolamellarin a, pyrrole derivative, rhodium, unclassified drug, neolamellarin A, triazole derivative, annulation reaction, antineoplastic activity, Article, cyclization, drug synthesis, reaction time, transannulation, catalysis, chemical structure, chemistry, synthesis, Pyrroles, Organic reaction, Present method, medicine, Organic chemistry, medicine.drug
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12Academic Journal
المصدر: Cohrt , A E OH , Le Quement , S T & Nielsen , T E 2014 , ' Solid-phase synthesis of NH-1,2,3-triazoles using 4,4′- bismethoxybenzhydryl azide ' , Synlett , vol. 25 , no. 13 , pp. 1891-1895 . https://doi.org/10.1055/s-0034-1378228
مصطلحات موضوعية: Organic Chemistry, azide, click chemistry, cross-coupling, N H-1,2,3-triazoles, solid-phase synthesis, 1,2,3 triazole derivative, 4,4' bismethoxybenzhydryl azide, alkyne derivative, unclassified drug, article, chemical structure, cycloaddition, deprotection reaction, reaction analysis, solid phase synthesis, stoichiometry
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13Academic Journal
المؤلفون: Doiron, J., Soultan, A.H., Richard, R., Touré, M.M., Picot, N., Čuperlović-Culf, M., Robichaud, G.A., Touaibia, M.
مصطلحات موضوعية: 1 (4 cyanophenylmethyl) 1h 1,2,3 triazole, 1 (4 cyanophenylmethyl) 1h imidazole, 1 (4,4' dicyanodiphenylmethyl) 1h 1,2,3 triazole, 1 (4,4' dicyanodiphenylmethyl) 1h imidazole, 1 (4,4' dicyanodiphenylmethyl) 4 [(4 cyanophenoxy)methyl] 1h 1,2,3 triazole, 1 (4,4' dicyanodiphenylmethyl) 4 hexyl 1h 1,2,3 triazole, 1 (4,4' dicyanodiphenylmethyl) 4 propyl 1h 1,2,3 triazole, 1 (diphenylmethyl) 1h imidazole, 1 (phenylmethyl) 4 cyano phenoxymethyl 1h 1,2,3 triazole, 1 (phenylmethyl) 4 methyl phenoxymethyl 1h 1,2,3 triazole, 1 (phenylmethyl) 4 nitro phenoxymethyl 1h 1,2,3 triazole, 1,2,3 triazole derivative, 1,2,5 triazole derivative, 2 (4,4' dicyanodiphenylmethyl) 2h 1,2,3 triazole, aromatase inhibitor, letrozole, triazole derivative, unclassified drug, adrenal cortex carcinoma, cancer growth, carcinoma cell, drug binding, drug inhibition, drug screening, drug structure, drug synthesis, human cell, IC 50, in vitro study, structure activity relation
وصف الملف: text
Relation: European Journal of Medicinal Chemistry, Volume: 46, Issue: 9, Publication date: 2011, Pages: 4010–4024
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14Academic Journal
المؤلفون: Tsyrenova B., Khrustalev V., Nenajdenko V.
المصدر: Journal of Organic Chemistry
مصطلحات موضوعية: Emission spectroscopy, Absorption and emission spectra, Heterocyclic systems, Isoquinoline ring, Photophysical properties, Photophysical studies, Steric hindrances, Synthetic strategies, Three-step synthesis, Synthesis (chemical), 1,2,3 triazole derivative, isoquinoline derivative, Article, cyclization, cycloaddition, hydrogen bond, quantum yield, reaction analysis, Sonogashira reaction, spectrofluorometry, stereospecificity, substitution reaction, synthesis, X ray diffraction
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15Academic Journal
المؤلفون: Tatevosyan S.S., Kotovshchikov Y.N., Latyshev G.V., Erzunov D.A., Sokolova D.V., Beletskaya I.P., Lukashev N.V.
المصدر: Journal of Organic Chemistry
مصطلحات موضوعية: Cesium compounds, Sulfur compounds, Transition metals, 1 ,3-Dipolarcycloaddition, Deoxycholic acid, DFT calculation, Direct approach, Heterocycles, Metal-free conditions, Natural compounds, Triazole ring, Cyclization, antiinflammatory agent, antimalarial agent, antineoplastic agent, antivirus agent, deoxycholic acid derivative, dioxane, sulfonamide, sulfonamide tethered 5 iodo 1,2,3 triazole derivative, transition element, triazole derivative, unclassified drug, annulation reaction, Article, chemical modification, cycloaddition, density functional theory, drug structure
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16Academic Journal
المؤلفون: Berrino E., Angeli A., Zhdanov D.D., Kiryukhina A.P., Milaneschi A., Bozdag M., Carradori S., Selleri S., Bartolucci G., Peat T.S., Ferraroni M., Supuran C.T., Carta F., De Luca A.
المصدر: Journal of Medicinal Chemistry
مصطلحات موضوعية: 1 [4 [4 [[(2,2 dioxidobenzo[e][1,2]oxathiin 6 yl)oxy]methyl] 1h 1,2,3 triazol 1 yl] 5 (hydroxymethyl)tetrahydrofuran 2 yl] 5 methylpyrimidine 2,4(1h,3h)dione, 1 [5 (hydroxymethyl) 4 [4 [3 [(2 oxo 2h chromen 6 yl)oxy]propyl] 1h 1,2,3 triazol 1 yl]tetrahydrofuran 2 yl] 5 methylpyrimidine 2,4(1h,3h)dione, 1 [5 (hydroxymethyl) 4 [4 [3 [(2 oxo 2h chromen 7 yl)oxy]propyl] 1h 1,2,3 triazol 1 yl]tetrahydrofuran 2 yl] 5 methylpyrimidine 2,4(1h,3h)dione, 1 [5 (hydroxymethyl) 4 [4 [4 [(2 oxo 2h chromen 4 yl)oxy]butyl] 1h 1,2,3 triazol 1 yl]tetrahydrofuran 2 yl] 5 methylpyrimidine 2,4(1h,3h)dione, 1 [5 (hydroxymethyl) 4 [4 [4 [(2 oxo 2h chromen 7 yl)oxy]butyl] 1h 1,2,3 triazol 1 yl]tetrahydrofuran 2 yl] 5 methylpyrimidine 2,4(1h,3h)dione, 1 [5 (hydroxymethyl) 4 [4 [[(2 oxo 2h chromen 6 yl)oxy]methyl] 1h 1,2,3 triazol 1 yl]tetrahydrofuran 2 yl] 5 methylpyrimidine 2,4(1h,3h)dione, 1 [5 (hydroxymethyl) 4 [4 [[(2 oxo 2h chromen 7 yl)oxy]methyl] 1h 1,2,3 triazol 1 yl]tetrahydrofuran 2 yl] 5 methylpyrimidine 2,4(1h,3h)dione, 1,2,3 triazole derivative, 3 [3 [4 [[[1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methyl]selanyl]phenyl]thioureido]benzenesulfonamide, 3 [3 [[1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methyl]ureido]benzenesulfonamide, 3 [[1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methyl] 2 oxo 2,3 dihydrobenzo[d]oxazole 5 sulfonamide, 4 [2 [bis[[1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methyl]amino]ethyl]benzenesulfonamide, 4 [3 [4 [[[1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methyl]selanyl]phenyl]thioureido]benzenesulfonamide, 4 [3 [[1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methyl]ureido]benzenesulfonamide, 4 [bis[[1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methyl]amino]benzenesulfonamide, 4 [[1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methoxy]benzenesulfonamide, 4 [[[1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methyl]amino]benzenesulfonamide, 4 [[[1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methyl]thio]benzenesulfonamide, acetazolamide, carbonate dehydratase inhibitor, carbonate dehydratase IX, carbonate dehydratase XII, n [[1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methyl] 4 sulfamoylbenzamide, telomerase inhibitor, unclassified drug, zidovudine, [1 [2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl] 1h 1,2,3 triazol 4 yl]methyl 4 sulfamoylbenzoate, [1 [[2 (hydroxymethyl) 5 (5 methyl 2,4 dioxo 3,4 dihydropyrimidin 1(2h)yl)tetrahydrofuran 3 yl]methyl] 1h 1,2,3 triazol 4 yl]methyl 4 chloro 3 sulfamoylbenzoate, antineoplastic activity, Article