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1
المؤلفون: Janet Lineberger, Emilio A. Emini, Julie A. DeMartino, Dooseop Kim, Michael W. Miller, Richard J. Budhu, Karen Henry, Renee Hrin, Gwen Carver, Lorraine Malkowitz, Anthony Carella, William A. Schleif, Malcolm MacCoss, Sandra L. Gould, Joseph Kessler, Daria J. Hazuda, Sander G. Mills, Christopher L. Lynch, Liping Wang, Jeffrey J. Hale, Martin S. Springer
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:2129-2134
مصطلحات موضوعية: Imidazopyridine, Pyrrolidines, Receptors, CCR5, Anti-HIV Agents, Stereochemistry, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, CCR5 receptor antagonist, Biochemistry, Pyrrolidine, chemistry.chemical_compound, Heterocyclic Compounds, Drug Discovery, Side chain, Animals, Humans, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Antagonist, virus diseases, Biological activity, Rats, CCR5 Receptor Antagonists, Molecular Medicine, Piperidine, HeLa Cells
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2
المؤلفون: Renee Danzeisen, Joseph Kessler, Karen Holmes, Anthony Carella, Janet Lineberger, Martin S. Springer, Malcolm MacCoss, Daria J. Hazuda, Natalie Chen, Sander G. Mills, Julie A. DeMartino, Emilio A. Emini, William A. Schleif, Gwen Carver, Shrenik K. Shah, Ravindra N. Guthikonda, Sandra L. Gould, Michael W. Miller, Lorraine Malkowitz
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:977-982
مصطلحات موضوعية: Anti-HIV Agents, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, CCR5 receptor antagonist, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Drug Discovery, Moiety, Sulfones, Molecular Biology, Dose-Response Relationship, Drug, Bicyclic molecule, Organic Chemistry, Antagonist, virus diseases, Butane, In vitro, chemistry, CCR5 Receptor Antagonists, Viruses, Butanes, Molecular Medicine, Piperidine
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3
المؤلفون: Karen Holmes, Emilio A. Emini, Karla L. Donnelly, Daria J. Hazuda, Sander G. Mills, Sandra L. Gould, Joseph Kessler, Malcolm MacCoss, William A. Schleif, Shrenik K. Shah, Ravindra N. Guthikonda, Janet Lineberger, Michael D. Miller, Salvatore J. Siciliano, Anthony Carella, Gwen Carver, Martin S. Springer, Kothandaraman Shankaran, Lorraine Malkowitz
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:3419-3424
مصطلحات موضوعية: Pyrrolidines, Anti-HIV Agents, Stereochemistry, Carboxylic acid, Clinical Biochemistry, Pharmaceutical Science, Acetates, Biochemistry, Chemical synthesis, HeLa, Structure-Activity Relationship, Chemokine receptor, Acetic acid, chemistry.chemical_compound, Piperidines, Drug Discovery, Humans, Structure–activity relationship, Binding site, Molecular Biology, chemistry.chemical_classification, Binding Sites, biology, Organic Chemistry, virus diseases, biology.organism_classification, In vitro, chemistry, CCR5 Receptor Antagonists, HIV-1, Molecular Medicine, Cell Division, HeLa Cells
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4
المؤلفون: Kevin T. Chapman, Jerry Di Salvo, Gloria Y. Kwei, Salvatore J. Siciliano, Dong-Ming Shen, Min Shu, Janet Lineberger, Kathy Lyons, Gwen Carver, Karen Holmes, Renee Danzeisen, Jennifer L. Loebach, Joseph Kessler, Martin S. Springer, James V. Pivnichny, Lorraine Malkowitz, Kerry A Parker, William A. Schleif, Emilio A. Emini, Daria J. Hazuda, Sander G. Mills, Sandra L. Gould, Anthony Carella, Julie A. DeMartino, Michael D. Miller
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:947-952
مصطلحات موضوعية: Anti-HIV Agents, Stereochemistry, Clinical Biochemistry, Substituent, Biological Availability, Pharmaceutical Science, CCR5 receptor antagonist, Biochemistry, Chemical synthesis, Monocytes, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Piperidines, Drug Discovery, Animals, Humans, Structure–activity relationship, Molecular Biology, Molecular Structure, Chemistry, Organic Chemistry, Rats, CCR5 Receptor Antagonists, Alkoxy group, Benzyl group, Pyrazoles, Molecular Medicine, Piperidine, Selectivity, HeLa Cells
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5
المؤلفون: Min Shu, Janet Lineberger, William A. Schleif, Salvatore J. Siciliano, Renee Danzeisen, Joseph Kessler, Karen Holmes, Martin S. Springer, Julie A. DeMartino, Kevin T. Chapman, Dong-Ming Shen, Anthony Carella, Lorraine Malkowitz, Michael D. Miller, Gloria Y. Kwei, Daria J. Hazuda, Sander G. Mills, Emilio A. Emini, Gwen Carver, Sandra L. Gould
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:935-939
مصطلحات موضوعية: Anti-HIV Agents, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Pyrazole, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Drug Discovery, Side chain, Animals, Humans, Moiety, Phenyl group, Isoxazole, Molecular Biology, Molecular Structure, Organic Chemistry, Rats, chemistry, CCR5 Receptor Antagonists, Benzyl group, Pyrazoles, Molecular Medicine, Piperidine, Cell Division, HeLa Cells
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6
المؤلفون: Margaret A. Cascieri, Salvatore J. Siciliano, Karen Holmes, Sandra L. Gould, Kevin T. Chapman, William A. Schleif, J. J. Hale, Richard J. Budhu, Renee Danzeisen, Joseph Kessler, Anthony Carella, Julie A. DeMartino, Christopher A. Willoughby, Daria J. Hazuda, Sander G. Mills, Malcolm MacCoss, Michael W. Miller, Janet Lineberger, Emilio A. Emini, Lorraine Malkowitz, Keith G. Rosauer, Martin S. Springer, Gwen Carver
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:427-431
مصطلحات موضوعية: Pyrrolidines, Anti-HIV Agents, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, CCR5 receptor antagonist, Biochemistry, Chemical synthesis, Pyrrolidine, chemistry.chemical_compound, Piperidines, In vivo, Cricetinae, Drug Discovery, Side chain, Animals, Humans, Chemokine CCL4, Molecular Biology, Organic Chemistry, Antagonist, Hydrogen Bonding, Macrophage Inflammatory Proteins, In vitro, Rats, chemistry, CCR5 Receptor Antagonists, Molecular Medicine, Piperidine, Half-Life, HeLa Cells
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7
المؤلفون: Emilio A. Emini, Julie A. DeMartino, Salvatore J. Siciliano, Karen Holmes, Gwen Carver, Sandra L. Gould, Kevin T. Chapman, Anthony Carella, Renee Danzeisen, Michael W. Miller, Joseph Kessler, Malcolm MacCoss, Christopher L. Lynch, Daria J. Hazuda, Sander G. Mills, Janet Lineberger, Lorraine Malkowitz, Amy Gentry, Richard J. Budhu, Jeffrey J. Hale, William A. Schleif, Margaret A. Cascieri, Martin S. Springer
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:3001-3004
مصطلحات موضوعية: Cell Membrane Permeability, Pyrrolidines, Chemical Phenomena, Anti-HIV Agents, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, CCR5 receptor antagonist, Biochemistry, Chemical synthesis, Pyrrolidine, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Cricetinae, Drug Discovery, Animals, Humans, Structure–activity relationship, Chemokine CCL4, Molecular Biology, Chemistry, Physical, Chemistry, Chinese hamster ovary cell, Organic Chemistry, Antagonist, Macrophage Inflammatory Proteins, In vitro, Rats, CCR5 Receptor Antagonists, HIV-1, Molecular Medicine, Indicators and Reagents, HeLa Cells
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8
المؤلفون: Anthony Carella, Kevin T. Chapman, Christopher A. Willoughby, Martin S. Springer, Lorraine Malkowitz, Janet Lineberger, Emilio A. Emini, Karen Holmes, Keith G. Rosauer, Scott C. Berk, Gwen Carver, Michael W. Miller, Silvia Degrado, Sandra L. Gould, Daria J. Hazuda, Renee Danzeisen, Joseph Kessler, William A. Schleif
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:3137-3141
مصطلحات موضوعية: Library design, Combinatorial Chemistry Techniques, biology, Chemistry, Chemokine receptor CCR5, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Antagonist, virus diseases, Pharmaceutical Science, CCR5 receptor antagonist, Combinatorial synthesis, Biochemistry, Chemical synthesis, Structure-Activity Relationship, CCR5 Receptor Antagonists, Drug Discovery, HIV-1, biology.protein, Molecular Medicine, Structure–activity relationship, Molecular Biology
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9
المؤلفون: William A. Schleif, Karen Holmes, Julie A. DeMartino, Liping Wang, Anthony Carella, Gwen Carver, Lorraine Malkowitz, Malcolm MacCoss, Paul E. Finke, Bryan Oates, Janet Lineberger, Emilio A. Emini, Ping Chen, Renee Danzeisen, Joseph Kessler, Michael W. Miller, Martin S. Springer, Sandra L. Gould, Daria J. Hazuda, Sander G. Mills, Dooseop Kim, Charles G. Caldwell
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:3099-3102
مصطلحات موضوعية: Anti-HIV Agents, Chemokine receptor CCR5, Clinical Biochemistry, Human immunodeficiency virus (HIV), Pharmaceutical Science, HIV Infections, Pharmacology, medicine.disease_cause, Biochemistry, Chemical synthesis, Virus, Drug Discovery, medicine, Humans, skin and connective tissue diseases, Molecular Biology, biology, Chemistry, Hydantoins, fungi, Organic Chemistry, biology.organism_classification, In vitro, body regions, CCR5 Receptor Antagonists, Lentivirus, Benzene derivatives, HIV-1, Hydantoin derivatives, biology.protein, Molecular Medicine
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10
المؤلفون: Janet Lineberger, Julie A. DeMartino, Salvatore J. Siciliano, Paul E. Finke, Richard J. Budhu, Gwen Carver, Malcolm MacCoss, Karen Holmes, Jeffrey J. Hale, Renee Danzeisen, Sandra L. Gould, Joseph Kessler, Bryan Oates, Edward Holson, William A. Schleif, Anthony Carella, Emilio A. Emini, Daria J. Hazuda, Sander G. Mills, Lorraine Malkowitz, Michael W. Miller, Martin S. Springer
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:2741-2745
مصطلحات موضوعية: Pyrrolidines, Anti-HIV Agents, Stereochemistry, Clinical Biochemistry, Nitro compound, Administration, Oral, Biological Availability, Pharmaceutical Science, CHO Cells, Microbial Sensitivity Tests, CCR5 receptor antagonist, Biochemistry, Chemical synthesis, Pyrrolidine, Structure-Activity Relationship, chemistry.chemical_compound, Oral administration, Cricetinae, Drug Discovery, Animals, Humans, Molecular Biology, chemistry.chemical_classification, biology, Organic Chemistry, Antagonist, HIV, virus diseases, biology.organism_classification, In vitro, chemistry, CCR5 Receptor Antagonists, Lentivirus, Molecular Medicine, HeLa Cells
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11
المؤلفون: Paul E. Finke, Emilio A. Emini, Sandra L. Gould, Michael W. Miller, Martin S. Springer, Lorraine Malkowitz, Anthony Carella, Karen Holmes, Julie A. DeMartino, Gwen Carver, Daria J. Hazuda, Sander G. Mills, Renee Danzeisen, Joseph Kessler, William A. Schleif, Malcolm MacCoss, Janet Lineberger, Bryan Oates
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:2475-2479
مصطلحات موضوعية: Anti-HIV Agents, Neutrophils, Stereochemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, CCR5 receptor antagonist, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Cricetinae, Drug Discovery, Animals, Humans, Structure–activity relationship, Molecular Biology, IC50, Cells, Cultured, Alkyl, chemistry.chemical_classification, Organic Chemistry, Antagonist, chemistry, Drug Design, CCR5 Receptor Antagonists, Butanes, HIV-1, Molecular Medicine, Piperidine, Selectivity
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12
المؤلفون: Karen Holmes, Michael W. Miller, Malcolm MacCoss, Lorraine Malkowitz, Renee Danzeisen, Gwen Carver, Salvatore J. Siciliano, Martin S. Springer, Joseph Kessler, Daria J. Hazuda, Sander G. Mills, Julie A. DeMartino, Bruce L. Daugherty, Janet Lineberger, William A. Schleif, Emilio A. Emini, Bryan Oates, Anthony Carella, Laura C. Meurer, Sandra L. Gould, Paul E. Finke
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:265-270
مصطلحات موضوعية: Anti hiv 1, Receptors, CCR5, Anti-HIV Agents, Stereochemistry, Chemokine receptor CCR5, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, CCR5 receptor antagonist, Butylamines, Transfection, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Cricetinae, Drug Discovery, Animals, Combinatorial Chemistry Techniques, Humans, Chemokine CCL4, Molecular Biology, IC50, Sulfonamides, biology, Aryl, Organic Chemistry, Butane, Macrophage Inflammatory Proteins, chemistry, CCR5 Receptor Antagonists, Butanes, Lead structure, biology.protein, Molecular Medicine, Antagonism, Protein Binding
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13
المؤلفون: Karen Holmes, Charles G. Caldwell, Salvatore J. Siciliano, Renee Danzeisen, Joseph Kessler, Julie A. DeMartino, Martin S. Springer, Ping Chen, William A. Schleif, Shrenik K. Shah, Michael D. Miller, Daria J. Hazuda, Sander G. Mills, Gwen Carver, Kothandaraman Shankaran, Malcolm MacCoss, Janet Lineberger, Lorraine Malkowitz, Karla L. Donnelly, Anthony Carella, Sandra L. Gould, Emilio A. Emini, Paul E. Finke, Gloria Kwei, Bryan Oates
المصدر: Bioorganicmedicinal chemistry letters. 14(13)
مصطلحات موضوعية: Receptors, CCR5, Stereochemistry, Anti-HIV Agents, Clinical Biochemistry, Human immunodeficiency virus (HIV), Pharmaceutical Science, medicine.disease_cause, Biochemistry, Chemical synthesis, Sulfone, Cell Line, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, Piperidines, Drug Discovery, medicine, Humans, Sulfones, Molecular Biology, Biological evaluation, Binding Sites, Chemistry, Organic Chemistry, virus diseases, Stereoisomerism, Cd4 receptors, In vitro, Drug Design, Benzene derivatives, CCR5 Receptor Antagonists, CD4 Antigens, Molecular Medicine, Piperidine
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14
المؤلفون: Salvatore J. Siciliano, Karen Holmes, Jeffrey J. Hale, Dong-Ming Shen, Shrenik K. Shah, Christopher A. Willoughby, Michael D. Miller, Anthony Carella, Lorraine Malkowitz, Julie A. DeMartino, Kathy Lyons, Min Shu, James V. Pivnichny, Emilio A. Emini, William A. Schleif, Gloria Y. Kwei, Martin S. Springer, Gwen Carver, Renee Danzeisen, Sandra L. Gould, Joseph Kessler, Daria J. Hazuda, Sander G. Mills, Christopher L. Lynch, Janet Lineberger, Kevin T. Chapman
المصدر: Bioorganicmedicinal chemistry letters. 14(4)
مصطلحات موضوعية: Anti-HIV Agents, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Biological Availability, Pyrazole, Acetates, Biochemistry, Chemical synthesis, Pyrrolidine, Monocytes, chemistry.chemical_compound, Acetic acid, Structure-Activity Relationship, Dogs, Piperidines, Pyrazole Compound, Drug Discovery, Organic chemistry, Animals, Humans, Molecular Biology, Molecular Structure, Organic Chemistry, Combinatorial chemistry, Macaca mulatta, Rats, chemistry, CCR5 Receptor Antagonists, Molecular Medicine, Pyrazoles, Piperidine, Trifluoromethanesulfonate, Isopropyl, HeLa Cells
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15
المؤلفون: Kevin T. Chapman, Karen Holmes, Salvatore J. Siciliano, Gwen Carver, Michael W. Miller, Julie A. DeMartino, Malcolm MacCoss, Margaret A. Cascieri, Richard J. Budhu, Emilio A. Emini, Paul E. Finke, Janet Lineberger, Daria J. Hazuda, Sander G. Mills, Lorraine Malkowitz, Anthony Carella, Dong-Ming Shen, Jeffrey J. Hale, Sandra L. Gould, Amy L. Gentry, Christopher L. Lynch, Charles G. Caldwell, Martin S. Springer, William A. Schleif, Renee Danzeisen, Joseph Kessler
المصدر: Organic letters. 5(14)
مصطلحات موضوعية: Anti hiv activity, Pyrrolidines, biology, Stereochemistry, Chemokine receptor CCR5, Anti-HIV Agents, Organic Chemistry, Biological Availability, Biochemistry, chemistry.chemical_compound, Pharmacokinetics, chemistry, CCR5 Receptor Antagonists, biology.protein, Physical and Theoretical Chemistry, Propionates, Cyclopentane
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16
المؤلفون: Christopher L. Lynch, Janet Lineberger, Julie A. DeMartino, Ping Chen, Scott C. Berk, Margaret A. Cascieri, Gwen Carver, Michael W. Miller, Edward J. Holson, Liya Chen, Martin S. Springer, Sandra L. Gould, Kevin T. Chapman, Jeffrey J. Hale, Karen Holmes, Renee Danzeisen, William A. Schleif, Malcolm MacCoss, Joseph Kessler, Richard J. Budhu, Anthony Carella, Charles G. Caldwell, Christopher A. Willoughby, Lorraine Malkowitz, Daria J. Hazuda, Sander G. Mills, Salvatore J. Siciliano, Emilio A. Emini, Amy Gentry, Keith G. Rosauer
المصدر: Bioorganicmedicinal chemistry letters. 13(1)
مصطلحات موضوعية: Pyrrolidines, Stereochemistry, Anti-HIV Agents, Metabolic Clearance Rate, Clinical Biochemistry, Pharmaceutical Science, CCR5 receptor antagonist, Biochemistry, Chemical synthesis, Pyrrolidine, Sulfone, chemistry.chemical_compound, Radioligand Assay, Structure-Activity Relationship, Dogs, Piperidines, Drug Discovery, Tumor Cells, Cultured, Moiety, Animals, Humans, Methylene, Molecular Biology, Organic Chemistry, Antagonist, Macaca mulatta, Rats, chemistry, CCR5 Receptor Antagonists, Leukocytes, Mononuclear, Molecular Medicine, Piperidine, Half-Life
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17
المؤلفون: Gwen Carver, Lorraine Malkowitz, Michael W. Miller, Karen Holmes, Salvatore J. Siciliano, Jeffrey J. Hale, Daria J. Hazuda, Martin S. Springer, Sander G. Mills, Julie A. DeMartino, Renee Danzeisen, Joseph Kessler, Malcolm MacCoss, Janet Lineberger, William A. Schleif, Richard J. Budhu, Sandra L. Gould, Anthony Carella, Emilio A. Emini
المصدر: Bioorganicmedicinal chemistry letters. 12(20)
مصطلحات موضوعية: Anti hiv 1, Calcium Channels, L-Type, Chemical Phenomena, Receptors, CCR5, Stereochemistry, Anti-HIV Agents, Clinical Biochemistry, Pharmaceutical Science, CCR5 receptor antagonist, CHO Cells, Biochemistry, Chemical synthesis, Pyrrolidine, chemistry.chemical_compound, Structure-Activity Relationship, Cricetinae, Drug Discovery, Animals, Humans, Chemokine CCL4, Molecular Biology, Chemistry, Chemistry, Physical, Calcium channel, Organic Chemistry, Antagonist, virus diseases, Macrophage Inflammatory Proteins, In vitro, Rats, CCR5 Receptor Antagonists, HIV-1, Molecular Medicine, Selectivity, Half-Life, HeLa Cells
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18
المؤلفون: Anthony Carella, Martin S. Springer, Margaret A. Cascieri, Emilio A. Emini, Lorraine Malkowitz, Malcolm MacCoss, Janet Lineberger, Sandra L. Gould, Karen Holmes, Daria J. Hazuda, Sander G. Mills, George A. Doss, Julie A. DeMartino, Michael W. Miller, Salvatore J. Siciliano, Renee Danzeisen, Joseph Kessler, Christopher L. Lynch, Gwen Carver, Amy Gentry, William A. Schleif, Jeffrey J. Hale
المصدر: Bioorganicmedicinal chemistry letters. 12(4)
مصطلحات موضوعية: Pyrrolidines, Chemokine receptor CCR5, Stereochemistry, Anti-HIV Agents, Clinical Biochemistry, Human immunodeficiency virus (HIV), Molecular Conformation, Pharmaceutical Science, Microbial Sensitivity Tests, medicine.disease_cause, Biochemistry, Chemical synthesis, Nitrone, Structure-Activity Relationship, Drug Discovery, medicine, Humans, Molecular Biology, chemistry.chemical_classification, biology, Bicyclic molecule, Organic Chemistry, virus diseases, Isoxazoles, Bridged Bicyclo Compounds, Heterocyclic, Cycloaddition, chemistry, CCR5 Receptor Antagonists, biology.protein, HIV-1, Molecular Medicine, Pharmacophore, Protein Binding
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19
المؤلفون: Anthony Carella, Janet Lineberger, Karen Holmes, Julie A. DeMartino, Sandra L. Gould, Liping Wang, Ping Chen, Paul E. Finke, Gwen Carver, Daria J. Hazuda, Sander G. Mills, Michael W. Miller, William A. Schleif, Martin S. Springer, Emilio A. Emini, Bryan Oates, Renee Danzeisen, Lorraine Malkowitz, Malcolm MacCoss, Joseph Kessler, Charles G. Caldwell, Dooseop Kim
المصدر: Bioorganicmedicinal chemistry letters. 11(24)
مصطلحات موضوعية: Stereochemistry, Chemokine receptor CCR5, Anti-HIV Agents, Clinical Biochemistry, Human immunodeficiency virus (HIV), Pharmaceutical Science, Hydantoin, HIV Infections, medicine.disease_cause, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Heterocyclic Compounds, Drug Discovery, medicine, Moiety, Humans, Molecular Biology, biology, Bicyclic molecule, Organic Chemistry, Antagonist, In vitro, chemistry, CCR5 Receptor Antagonists, biology.protein, HIV-1, Molecular Medicine, HeLa Cells
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20
المؤلفون: Janet Lineberger, Salvatore J. Siciliano, Michael W. Miller, Karen Holmes, Lorraine Malkowitz, Renee Danzeisen, Richard J. Budhu, Joseph Kessler, Conrad P. Dorn, Julie A. DeMartino, Malcolm MacCoss, Gwen Carver, Bruce L. Daugherty, William A. Schleif, Bryan Oates, Martin S. Springer, Emilio A. Emini, Paul E. Finke, Daria J. Hazuda, Sander G. Mills, Anthony Carella, Sandra L. Gould
المصدر: Bioorganicmedicinal chemistry letters. 11(2)
مصطلحات موضوعية: Receptors, CCR5, Chemokine receptor CCR5, Stereochemistry, Anti-HIV Agents, Clinical Biochemistry, Pharmaceutical Science, CCR5 receptor antagonist, CHO Cells, Transfection, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, Piperidines, Cricetinae, Drug Discovery, Structure–activity relationship, Animals, Combinatorial Chemistry Techniques, Humans, Chemokine CCL4, Molecular Biology, chemistry.chemical_classification, biology, Organic Chemistry, Benzothiophene, Sulfoxide, Macrophage Inflammatory Proteins, Sulfonamide, chemistry, CCR5 Receptor Antagonists, biology.protein, Molecular Medicine, Sample collection, Protein Binding